| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4385789 | A | Inhibition of PDE1B catalytic domain (10 to 487 residues) (unknown origin) using 3H-cGMP as substrate after 15 mins by liquid scintillation counting method | Homo sapiens | 15 | single protein format | Scientific Literature | ||
| 2. | ALA4385790 | B | Selectivity ratio of IC50 for PDE1B catalytic domain (10 to 487 residues) (unknown origin) to IC50 for recombinant human PDE9A2 catalytic domain (181 to 506 residues) expressed in Escherichia coli BL21 | Homo sapiens | 14 | assay format | Scientific Literature | ||
| 3. | ALA4385793 | A | Half life in rat liver microsomes at 1.5 uM | Rattus norvegicus | 3 | microsome format | Scientific Literature | ||
| 4. | ALA4385795 | A | Hepatic extraction ratio in rat liver microsomes at 1.5 uM | Rattus norvegicus | 3 | microsome format | Scientific Literature | ||
| 5. | ALA4385797 | A | Stability in rat liver microsomes assessed as stability constant at 1.5 uM | Rattus norvegicus | 3 | microsome format | Scientific Literature | ||
| 6. | ALA4385798 | A | Intrinsic clearance in rat liver microsomes at 1.5 uM | Rattus norvegicus | 3 | microsome format | Scientific Literature | ||
| 7. | ALA4385799 | A | Apparent clearance in rat liver microsomes at 1.5 uM | Rattus norvegicus | 3 | microsome format | Scientific Literature | ||
| 8. | ALA4385800 | A | Hepatic clearance in rat liver microsomes at 1.5 uM | Rattus norvegicus | 3 | microsome format | Scientific Literature | ||
| 9. | ALA4385807 | B | Inhibition of recombinant human PDE9A2 catalytic domain (181 to 506 residues) expressed in Escherichia coli BL21 using 3H-cGMP as substrate after 15 mins by liquid scintillation counting method | Homo sapiens | 14 | assay format | Scientific Literature |
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