# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4426351 | B | Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK293 cells by microbeta liquid scintillation counting | Homo sapiens | 28 | ALA4425120 | cell-based format | Scientific Literature | |
2. | ALA4426352 | B | Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells by microbeta liquid scintillation counting | Homo sapiens | 5 | ALA4425120 | cell-based format | Scientific Literature | |
3. | ALA4426353 | B | Displacement of [3H]-Ketanserin from human 5-HT2A receptor expressed in HEK293 cells by microbeta liquid scintillation counting | Homo sapiens | 5 | ALA4425120 | cell-based format | Scientific Literature | |
4. | ALA4426354 | B | Displacement of [3H]-5-CT from human 5-HT7B receptor expressed in HEK293 cells by microbeta liquid scintillation counting | Homo sapiens | 5 | ALA4425120 | cell-based format | Scientific Literature | |
5. | ALA4426355 | B | Displacement of [3H]-Raclopride from human D2L receptor expressed in HEK293 cells by microbeta liquid scintillation counting | Homo sapiens | 5 | ALA4425120 | cell-based format | Scientific Literature | |
6. | ALA4426356 | B | Selectivity ratio of Ki for human 5-HT1A receptor expressed in HEK293 cells to Ki for human 5-HT6 receptor expressed in HEK293 cells | Homo sapiens | 5 | ALA4425120 | cell-based format | Scientific Literature | |
7. | ALA4426357 | B | Selectivity ratio of Ki for human 5-HT2A receptor expressed in HEK293 cells to Ki for human 5-HT6 receptor expressed in HEK293 cells | Homo sapiens | 5 | ALA4425120 | cell-based format | Scientific Literature | |
8. | ALA4426358 | B | Selectivity ratio of Ki for human 5-HT7B receptor expressed in HEK293 cells to Ki for human 5-HT6 receptor expressed in HEK293 cells | Homo sapiens | 5 | ALA4425120 | cell-based format | Scientific Literature | |
9. | ALA4426359 | B | Selectivity ratio of Ki for human D2L receptor expressed in HEK293 cells to Ki for human 5-HT6 receptor expressed in HEK293 cells | Homo sapiens | 5 | ALA4425120 | cell-based format | Scientific Literature | |
10. | ALA4426360 | F | Antagonist activity at human recombinant 5-HT6 receptor expressed in CHO cells assessed as inhibition of serotonin-induced intracellular cAMP accumulation after 30 mins by HTRF assay | Homo sapiens | 2 | ALA4425120 | cell-based format | Scientific Literature | |
11. | ALA4426361 | B | Displacement of [3H]prazosin from rat cerebral cortex adrenergic alpha 1 receptor after 60 mins by scintillation counting | Rattus norvegicus | 2 | ALA4425120 | assay format | Scientific Literature | |
12. | ALA4426362 | B | Displacement of [3H]RX 821002 from human recombinant adrenergic alpha 2C receptor expressed in CHO cells after 60 mins by scintillation counting | Homo sapiens | 2 | ALA4425120 | cell-based format | Scientific Literature | |
13. | ALA4426363 | B | Displacement of [3H]pirenzepine from human recombinant muscarinic M1 receptor expressed in CHO cells after 60 mins by scintillation counting | Homo sapiens | 2 | ALA4425120 | cell-based format | Scientific Literature | |
14. | ALA4426364 | B | Displacement of [3H]4-DAMP from human recombinant muscarinic M5 receptor expressed in CHO cells after 60 mins by scintillation counting | Homo sapiens | 2 | ALA4425120 | cell-based format | Scientific Literature | |
15. | ALA4426365 | B | Displacement of [3H]mesulergine from human recombinant 5-HT2C receptor expressed in HEK293 cells after 120 mins by scintillation counting | Homo sapiens | 2 | ALA4425120 | cell-based format | Scientific Literature | |
16. | ALA4426366 | B | Displacement of [3H]imipramine from human recombinant SERT expressed in CHO cells after 60 mins by scintillation counting | Homo sapiens | 2 | ALA4425120 | cell-based format | Scientific Literature | |
17. | ALA4426367 | F | Agonist activity at human recombinant 5-HT2B receptor expressed in HEK-293 cells assessed as IP1 accumulation at 1 uM after 30 mins by HTRF assay | Homo sapiens | 2 | ALA4425120 | cell-based format | Scientific Literature | |
18. | ALA4426368 | B | Displacement of [3H]Dofetilide from human recombinant ERG expressed in HEK293 cells at 10 to 50 uM after 60 mins by scintillation counting | Homo sapiens | 2 | ALA4425120 | cell-based format | Scientific Literature | |
19. | ALA4426369 | B | Displacement of [3H]-methyl-spiperone from human recombinant dopamine D3 receptor expressed in CHO cells after 60 mins by scintillation counting | Homo sapiens | 2 | ALA4425120 | cell-based format | Scientific Literature | |
20. | ALA4426370 | A | Inhibition of human CYP1A2 expressed in supersomes assessed as caffeine 3-N-demethylation after 15 mins by HPLC analysis | Homo sapiens | 2 | ALA4425120 | assay format | Scientific Literature |