| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4392119 | B | Displacement of [3H]-LSD from recombinant human 5HT7A receptor stably expressed in HEK cells measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 2. | ALA4392120 | F | Agonist activity at recombinant human D1 receptor expressed in HEK29T cells assessed as induction of stimulatory G-protein-mediated cAMP accumulation measured after 15 mins by Glosensor-based FLIPR assay | Homo sapiens | 44 | cell-based format | Scientific Literature | ||
| 3. | ALA4392121 | F | Agonist activity at recombinant human D1 receptor expressed in HEK29T cells assessed as induction of stimulatory G-protein-mediated cAMP accumulation measured after 15 mins by Glosensor-based FLIPR assay relative to dopamine | Homo sapiens | 44 | cell-based format | Scientific Literature | ||
| 4. | ALA4392122 | B | Agonist activity at recombinant C-terminal RLuc8-fused human D1 receptor expressed in HEK29T cells co-expressing N-terminal Venus-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment measured after 15 mins in presence of coelenterazine H by BRET assay | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
| 5. | ALA4392123 | B | Agonist activity at recombinant C-terminal RLuc8-fused human D1 receptor expressed in HEK29T cells co-expressing N-terminal Venus-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment measured after 15 mins in presence of coelenterazine H by BRET assay relative to dopamine | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
| 6. | ALA4392126 | F | Bias factor, transduction co-efficient for agonist activity at recombinant human D1 receptor expressed in HEK29T cells assessed as induction of stimulatory G-protein-mediated cAMP accumulation to agonist activity at recombinant C-terminal RLuc8-fused human D1 receptor expressed in HEK29T cells co-expressing N-terminal Venus-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 7. | ALA4392129 | B | Displacement of [3H]-SCH23390 from recombinant human D1 receptor transiently expressed in HEKT cells measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 8. | ALA4392130 | B | Displacement of [3H]-N-methylspiperone from recombinant human D2 receptor stably expressed in fibroblast cells measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 9. | ALA4392131 | B | Displacement of [3H]-N-methylspiperone from D3 receptor (unknown origin) measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 10. | ALA4392132 | B | Displacement of [3H]-N-methylspiperone from recombinant human D4 receptor stably expressed in HEK cells measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 11. | ALA4392133 | B | Displacement of [3H]-SCH23390 from recombinant human D5 receptor transiently expressed in HEKT cells measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 12. | ALA4392134 | B | Displacement of [3H]-QNB/[3H]-NMS from human muscarinic M1 receptor expressed in stable CHO cells after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 13. | ALA4392135 | B | Displacement of [3H]-U69593 from KOR (unknown origin) measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 14. | ALA4392136 | B | Displacement of [3H]-Way100635 from recombinant human 5HT1A receptor stably expressed in CHO cells measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 15. | ALA4392137 | B | Displacement of [3H]5-CT from recombinant human 5HT1B receptor stably expressed in HEK cells measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 16. | ALA4392138 | B | Displacement of [3H]5-CT from recombinant human 5HT1D receptor transiently expressed in HEKT cells measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 17. | ALA4392139 | B | Displacement of [3H]5-HT from recombinant human 5HT1E receptor stably expressed in HEK cells measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 18. | ALA4392140 | B | Displacement of [3H]-Ketanserin from 5HT2A receptor (unknown origin) measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 19. | ALA4392141 | B | Displacement of [3H]-LSD from recombinant human 5HT2B receptor stably expressed in HEK cells measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 20. | ALA4392142 | B | Displacement of [3H]GR65630 from recombinant human 5HT3 receptor transiently expressed in HEKT cells measured after 90 mins by microbeta scintillation counting method | Homo sapiens | 4 | cell-based format | Scientific Literature |
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