# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4374936 | B | Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl coenzyme A and N-terminal histone H4 peptide (sequence SGRGKGGKGLGKGGAKRHRKV-GGK-biotin) as substrate incubated for 60 mins by Alpha screen technology | Homo sapiens | 72 | ALA4373691 | cell-based format | Scientific Literature | |
2. | ALA4374938 | B | Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 15 uM acetyl coenzyme A and N-terminal histone H4 peptide (sequence SGRGKGGKGLGKGGAKRHRKV-GGK-biotin) as substrate incubated for 60 mins by Alpha screen technology | Homo sapiens | 30 | ALA4373691 | cell-based format | Scientific Literature | |
3. | ALA4404752 | B | Inhibition of N-terminal NusA-fused His6-tagged human KAT6A (507 to 778 residues) expressed in Escherichia coli BL21 (DE3) cells using 0.4 uM acetyl coenzyme A and N-terminal histone H4 peptide (sequence SGRGKGGKGLGKGGAKRHRKV-GGK-biotin) as substrate incubated for 60 mins by Alpha screen technology | Homo sapiens | 177 | ALA4402574 | cell-based format | Scientific Literature | |
4. | ALA4407092 | B | Inhibition of KAT7 (unknown origin) | Homo sapiens | 1 | ALA4406797 | single protein format | Scientific Literature | |
5. | ALA4407093 | B | Inhibition of KAT5 (unknown origin) | Homo sapiens | 1 | ALA4406797 | single protein format | Scientific Literature | |
6. | ALA4407094 | B | Inhibition of KAT7 (unknown origin) assessed as reduction in H3K14ac acetylation at 10 uM relative to control | Homo sapiens | 1 | ALA4406797 | single protein format | Scientific Literature | |
7. | ALA4407095 | B | Inhibition of KAT7 (unknown origin) assessed as reduction in H3K9ac acetylation at 10 uM relative to control | Homo sapiens | 1 | ALA4406797 | single protein format | Scientific Literature |