| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4433975 | F | Agonist activity at human T1R2/T1R3 expressed in PEAKrapid cells assessed as effect on intracellular calcium influx measured for 120 secs by fluorescence based assay | Homo sapiens | 25 | cell-based format | Scientific Literature | ||
| 2. | ALA4433976 | F | Positive allosteric modulator activity at human T1R2/T1R3 expressed in PEAKrapid cells assessed as potentiation of sucrose-induced intracellular calcium influx by measuring sucrose EC50 at 30 uM measured for 120 secs by fluorescence based assay (Rvb = 31.7 mM) | Homo sapiens | 22 | cell-based format | Scientific Literature | ||
| 3. | ALA4433979 | F | Positive allosteric modulator activity at human T1R2/T1R3 expressed in PEAKrapid cells assessed as potentiation of sucrose-induced intracellular calcium influx by measuring sucrose EC50 at 30 uM measured for 120 secs by fluorescence based assay relative to FEMA4774 | Homo sapiens | 20 | cell-based format | Scientific Literature |
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