| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4312045 | Binding | Inhibition of BRD2 (unknown origin) by TR-FRET assay | Homo sapiens | 6 | ALA4311931 | single protein format | Scientific Literature | |
| 2. | ALA4312046 | Binding | Inhibition of BRD3 (unknown origin) by TR-FRET assay | Homo sapiens | 6 | ALA4311931 | single protein format | Scientific Literature | |
| 3. | ALA4312047 | Binding | Inhibition of BRD4 (unknown origin) by TR-FRET assay | Homo sapiens | 6 | ALA4311931 | single protein format | Scientific Literature | |
| 4. | ALA4312048 | Binding | Inhibition of BRD4 in human MX1 cells assessed as decrease in cell proliferation after 3 days by Celltiter-Glo assay | Homo sapiens | 6 | ALA4311931 | cell-based format | Scientific Literature | |
| 5. | ALA4312049 | Binding | Inhibition of BRD4 in human H1229 cells transfected with HPV-E2 assessed as transrepression of HPV-long control region by luciferase reporter assay | Homo sapiens | 6 | ALA4311931 | cell-based format | Scientific Literature | |
| 6. | ALA4312050 | ADME | Permeability of compound in 5% DMSO after 7 hrs by PAMPA | 40 | ALA4311931 | assay format | Scientific Literature | ||
| 7. | ALA4312051 | ADME | Ratio of drug concentration in unbound HEK293 cell to media | 13 | ALA4311931 | assay format | Scientific Literature | ||
| 8. | ALA4312074 | Binding | Inhibition of BRD4 in human MX1 cells assessed as decrease in cell proliferation after 3 days by Celltiter-Glo assay relative to parent compound | Homo sapiens | 5 | ALA4311931 | cell-based format | Scientific Literature | |
| 9. | ALA4312075 | Binding | Inhibition of BRD4 in luciferase expressing human H1229 cells transfected with HPV-E2 assessed as transrepression of HPV-long control region by luciferase reporter assay relative to parent compound | Homo sapiens | 5 | ALA4311931 | assay format | Scientific Literature |
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