| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4425261 | ADME | Binding affinity to wild type partial length human EGFR expressed in bacterial system by KINOMEscan assay | Homo sapiens | 7 | ALA4425085 | assay format | Scientific Literature | |
| 2. | ALA4425262 | Binding | Binding affinity to partial length human EGFR L858R/T790M double mutant expressed in mammalian system by KINOMEscan assay | Homo sapiens | 7 | ALA4425085 | assay format | Scientific Literature | |
| 3. | ALA4425263 | Binding | Selectivity ratio of Kd for wild type partial length human EGFR to Kd for partial length human EGFR L858R/T790M double mutant | Homo sapiens | 7 | ALA4425085 | assay format | Scientific Literature | |
| 4. | ALA4425264 | ADME | Antiproliferative activity against human A431 cells expressing wild type EGFR by MTS assay | Homo sapiens | 7 | ALA4425085 | cell-based format | Scientific Literature | |
| 5. | ALA4425265 | Functional | Antiproliferative activity against human NCI-H1975 cells expressing EGFR L858R/T790M double mutant by MTS assay | Homo sapiens | 7 | ALA4425085 | cell-based format | Scientific Literature | |
| 6. | ALA4425266 | Unassigned | Selectivity ratio of IC50 for human A431 cells expressing wild type EGFR to IC50 for human NCI-H1975 cells expressing EGFR L858R/T790M double mutant | Homo sapiens | 7 | ALA4425085 | assay format | Scientific Literature |
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