# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4337304 | Binding | Displacement of [3H]PK11195 from wild-type human TSPO expressed in HEK293 cell membranes after 90 mins by scintillation counting method | Homo sapiens | 30 | ALA4334481 | cell-based format | Scientific Literature | |
2. | ALA4337305 | Binding | Selectivity ratio of ki for human TSPO A147T mutant expressed in HEK293 cell membranes to ki for human TSPO expressed in HEK293 cell membranes | Homo sapiens | 19 | ALA4334481 | cell-based format | Scientific Literature | |
3. | ALA4337306 | Binding | Displacement of [3H]PK11195 from human TSPO A147T mutant expressed in HEK293 cell membranes after 90 mins by scintillation counting method | Homo sapiens | 30 | ALA4334481 | cell-based format | Scientific Literature | |
4. | ALA4337309 | Binding | Binding affinity to wild-type human TSPO expressed in HEK293 cells assessed as inhibition of cell viability at 100 uM incubated for 48 hrs by CellTiter Blue assay relative to control | Homo sapiens | 9 | ALA4334481 | cell-based format | Scientific Literature | |
5. | ALA4337310 | Binding | Binding affinity to human TSPO A147T mutant expressed in HEK293 cells assessed as inhibition of cell viability at 100 uM incubated for 48 hrs by CellTiter Blue assay relative to control | Homo sapiens | 9 | ALA4334481 | cell-based format | Scientific Literature | |
6. | ALA4337311 | Binding | Binding affinity to wild-type human TSPO expressed in HEK293 cells assessed as inhibition of cell proliferation at 100 uM incubated for 48 hrs by Brdu incorporation-based ELISA relative to control | Homo sapiens | 9 | ALA4334481 | cell-based format | Scientific Literature | |
7. | ALA4337312 | Binding | Binding affinity to human TSPO A147T mutant expressed in HEK293 cells assessed as inhibition of cell proliferation at 100 uM incubated for 48 hrs by Brdu incorporation-based ELISA relative to control | Homo sapiens | 9 | ALA4334481 | cell-based format | Scientific Literature |