| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4392940 | A | Renal clearance in dog | Canis lupus familiaris | 9 | assay format | Scientific Literature | ||
| 2. | ALA4392941 | A | Plasma clearance in dog | Canis lupus familiaris | 9 | assay format | Scientific Literature | ||
| 3. | ALA4392942 | B | Inhibition of recombinant human Kv1.5 expressed in CHO cells by IonWork high-throughput electrophysiology assay | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
| 4. | ALA4392943 | B | Inhibition of human ERG | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 5. | ALA4392944 | B | Inhibition of IKs (unknown origin) | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 6. | ALA4392950 | A | Drug metabolism in human hepatocytes assessed as glucuronidation | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 7. | ALA4392952 | A | Drug excretion in dog urine | Canis lupus familiaris | 9 | tissue-based format | Scientific Literature | ||
| 8. | ALA4392953 | B | Inhibition of Kv1.5 in human atrial myocytes assessed as blockade of Ikur current | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 9. | ALA4392954 | F | Antiarrhythmic activity in iv dosed anesthetized rabbit assessed as free compound plasma exposure which prolongs the right atrial effective refractory period by 20 milliseconds measured after 20 mins by electrophysiological analysis | Oryctolagus cuniculus | 4 | organism-based format | Scientific Literature | ||
| 10. | ALA4392955 | F | Antiarrhythmic activity in rapid atrial pacing dog model of atrial fibrillation assessed as unbound plasma concentration required to convert atrial fibrillation to sinus rhythm | Canis lupus familiaris | 1 | organism-based format | Scientific Literature | ||
| 11. | ALA4392957 | B | Inhibition of Kir3.1 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA4392958 | B | Inhibition of Kir3.4 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA4392959 | B | Inhibition of Kv4.3 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA4392960 | B | Inhibition of human ERG at 33 uM relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA4392961 | B | Inhibition of Nav1.5 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA4392962 | B | Inhibition of CaV1.2 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA4392963 | A | Proconvulsant activity in PTZ-induced rat model assessed as behavioral changes by Irwin test | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 18. | ALA4392964 | A | Free drug level in rat brain at 2 umol/kg/hr administered for 4 hrs | Rattus norvegicus | 1 | tissue-based format | Scientific Literature | ||
| 19. | ALA4392965 | B | Inhibition of NMDA receptor glycine binding site (unknown origin) at 10 uM relative to control | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 20. | ALA4392966 | B | Inhibition of NMDA receptor phencyclidine binding site (unknown origin) at 10 uM relative to control | Homo sapiens | 1 | protein complex format | Scientific Literature |
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