| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4427807 | Binding | Inhibition of human PRSS1 assessed as enzymatic cleavage of Benzoyl-GlyPro-Arg'Rh110-gammaGlu-OH by fluorescence analysis | Homo sapiens | 18 | ALA4425182 | single protein format | Scientific Literature | |
| 2. | ALA4427808 | Physicochemical | Dissociation constant, pKa of the compound | 4 | ALA4425182 | small-molecule physicochemical format | Scientific Literature | ||
| 3. | ALA4427809 | Binding | Displacement of [3H]-dofetilide from human ERG expressed in HEK293 cells measured after 90 mins by scintillation proximity assay | Homo sapiens | 14 | ALA4425182 | cell-based format | Scientific Literature | |
| 4. | ALA4427810 | Physicochemical | Solubility of the compound at pH 6.8 | 3 | ALA4425182 | small-molecule physicochemical format | Scientific Literature | ||
| 5. | ALA4427811 | ADME | Clearance in Sprague-Dawley rat at 1 mg/kg, iv | Rattus norvegicus | 2 | ALA4425182 | organism-based format | Scientific Literature | |
| 6. | ALA4427812 | ADME | AUC (0 to 24 hrs) in Sprague-Dawley rat at 1 mg/kg, iv | Rattus norvegicus | 2 | ALA4425182 | organism-based format | Scientific Literature | |
| 7. | ALA4427814 | Binding | Inhibition of human thrombin | Homo sapiens | 4 | ALA4425182 | single protein format | Scientific Literature | |
| 8. | ALA4427815 | Binding | Inhibition of human f10a | Homo sapiens | 4 | ALA4425182 | single protein format | Scientific Literature | |
| 9. | ALA4427816 | Binding | Inhibition of human neutrophil elastase | Homo sapiens | 4 | ALA4425182 | single protein format | Scientific Literature | |
| 10. | ALA4427817 | Binding | Inhibition of human chymotrypsin | Homo sapiens | 4 | ALA4425182 | protein format | Scientific Literature |
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