# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4395839 | Binding | Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISA | Homo sapiens | 39 | ALA4393708 | single protein format | Scientific Literature | |
2. | ALA4395841 | Binding | Competitive inhibition of human recombinant full length GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated with enzyme for 10 mins followed by substrate and 25 uM ATP addition measured after 60 mins by ADP-Glo luminescence assay | Homo sapiens | 40 | ALA4393708 | single protein format | Scientific Literature | |
3. | ALA4395842 | Binding | Inhibition of human recombinant full length GSK3alpha using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated with enzyme for 10 mins followed by substrate and 25 uM ATP addition measured after 60 mins by ADP-Glo luminescence assay | Homo sapiens | 6 | ALA4393708 | single protein format | Scientific Literature | |
4. | ALA4395846 | ADME | Metabolic stability in human liver microsomes assessed as parent compound remaining after 10 mins by LC-MS analysis relative to control | Homo sapiens | 3 | ALA4393708 | microsome format | Scientific Literature | |
5. | ALA4395847 | ADME | Metabolic stability in human liver microsomes assessed as parent compound remaining after 20 mins by LC-MS analysis relative to control | Homo sapiens | 3 | ALA4393708 | microsome format | Scientific Literature | |
6. | ALA4395848 | ADME | Metabolic stability in human liver microsomes assessed as parent compound remaining after 30 mins by LC-MS analysis relative to control | Homo sapiens | 3 | ALA4393708 | microsome format | Scientific Literature | |
7. | ALA4395849 | ADME | Metabolic stability in human liver microsomes assessed as parent compound remaining after 60 mins by LC-MS analysis relative to control | Homo sapiens | 3 | ALA4393708 | microsome format | Scientific Literature | |
8. | ALA4395850 | ADME | Metabolic stability in human liver microsomes assessed as parent compound remaining after 120 mins by LC-MS analysis relative to control | Homo sapiens | 3 | ALA4393708 | microsome format | Scientific Literature | |
9. | ALA4395851 | ADME | Metabolic stability in human liver microsomes assessed as parent compound remaining after 240 mins by LC-MS analysis relative to control | Homo sapiens | 4 | ALA4393708 | microsome format | Scientific Literature | |
10. | ALA4395866 | ADME | Metabolic stability in human liver microsomes assessed as parent compound remaining after 180 mins by LC-MS analysis relative to control | Homo sapiens | 3 | ALA4393708 | microsome format | Scientific Literature |