# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4430972 | Binding | Displacement of [3H]CCPA from human A1 receptor expressed in CHO cell membrane by liquid scintillation counting method | Homo sapiens | 12 | ALA4428125 | cell-based format | Scientific Literature | |
2. | ALA4430974 | Binding | Displacement of [3H]CCPA from A1 receptor in rat brain cortex membranes by liquid scintillation counting method | Rattus norvegicus | 61 | ALA4428125 | cell membrane format | Scientific Literature | |
3. | ALA4430980 | Binding | Displacement of [3H]MSX from A2A receptor in rat brain striatum membranes measured after 30 mins by liquid scintillation counting method | Rattus norvegicus | 62 | ALA4428125 | cell membrane format | Scientific Literature | |
4. | ALA4430981 | Binding | Displacement of [3H]MSX from human A2A receptor measured after 30 mins by liquid scintillation counting method | Homo sapiens | 8 | ALA4428125 | single protein format | Scientific Literature | |
5. | ALA4430983 | Binding | Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells preincubated for 30 mins followed by addition of p-tyramine as substrate measured over 45 mins by Amplex Red MAO assay | Homo sapiens | 65 | ALA4428125 | cell-based format | Scientific Literature | |
6. | ALA4430984 | Binding | Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells at 10 uM preincubated for 30 mins followed by addition of p-tyramine as substrate measured over 45 mins by Amplex Red MAO assay relative to control | Homo sapiens | 27 | ALA4428125 | cell-based format | Scientific Literature | |
7. | ALA4430985 | Binding | Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells preincubated for 30 mins followed by addition of p-tyramine as substrate measured over 45 mins by Amplex Red MAO assay | Homo sapiens | 65 | ALA4428125 | cell-based format | Scientific Literature | |
8. | ALA4430986 | Binding | Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells at 10 uM preincubated for 30 mins followed by addition of p-tyramine as substrate measured over 45 mins by Amplex Red MAO assay relative to control | Homo sapiens | 46 | ALA4428125 | cell-based format | Scientific Literature | |
9. | ALA4430992 | Binding | Displacement of [3H]PSB-603 from human A2B receptor expressed in CHO cell membrane | Homo sapiens | 63 | ALA4428125 | cell-based format | Scientific Literature | |
10. | ALA4430995 | Binding | Displacement of [3H]PSB-603 from human A2B receptor expressed in CHO cell membrane at 1 uM relative to control | Homo sapiens | 51 | ALA4428125 | cell-based format | Scientific Literature | |
11. | ALA4430997 | Binding | Displacement of [3H]PSB-11 from human A3 receptor expressed in CHO cell membrane by liquid scintillation counting method relative to control | Homo sapiens | 64 | ALA4428125 | cell-based format | Scientific Literature | |
12. | ALA4430998 | Binding | Displacement of [3H]PSB-11 from human A3 receptor expressed in CHO cell membrane at 10 uM by liquid scintillation counting method relative to control relative to control | Homo sapiens | 52 | ALA4428125 | cell-based format | Scientific Literature | |
13. | ALA4430999 | Physicochemical | Thermodynamic solubility of the compound at pH 1 | 25 | ALA4428125 | small-molecule physicochemical format | Scientific Literature | ||
14. | ALA4431000 | Physicochemical | Thermodynamic solubility of the compound at pH 4 | 25 | ALA4428125 | small-molecule physicochemical format | Scientific Literature | ||
15. | ALA4431001 | Physicochemical | Thermodynamic solubility of the compound at pH 7.4 | 25 | ALA4428125 | small-molecule physicochemical format | Scientific Literature |