# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4367878 | Binding | Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysis | Homo sapiens | 33 | ALA4364306 | cell-based format | Scientific Literature | |
2. | ALA4367879 | Binding | Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysis | Homo sapiens | 33 | ALA4364306 | cell-based format | Scientific Literature | |
3. | ALA4367880 | Binding | Selectivity index, ratio of Ki for recombinant human CB1R expressed in HEK293 cell membranes to Ki for recombinant human CB2R expressed in HEK293 cell membranes | Homo sapiens | 16 | ALA4364306 | cell-based format | Scientific Literature | |
4. | ALA4367881 | Binding | Agonist activity at N-terminal Flag epitope tagged CB2 (unknown origin) expressed in HTLA cells assessed as increase of beta-arrestin recruitment by Tango assay | Homo sapiens | 33 | ALA4364306 | cell-based format | Scientific Literature | |
5. | ALA4367882 | Binding | Antagonist activity at N-terminal Flag epitope tagged CB2 (unknown origin) expressed in HTLA cells assessed as decrease in CP55940-induced beta-arrestin recruitment pretreated with non-selective cannabinoid receptor agonist CP55940 for 30 mins and measured after 20 mins by Tango assay | Homo sapiens | 33 | ALA4364306 | cell-based format | Scientific Literature | |
6. | ALA4367883 | Binding | Agonist activity at N-terminal Flag epitope tagged CB1 (unknown origin) expressed in HTLA cells assessed as increase of beta-arrestin recruitment by Tango assay | Homo sapiens | 32 | ALA4364306 | cell-based format | Scientific Literature | |
7. | ALA4367884 | Binding | Antagonist activity at N-terminal Flag epitope tagged CB1 (unknown origin) expressed in HTLA cells assessed as decrease in CP55940-induced beta-arrestin recruitment pretreated with non-selective cannabinoid receptor agonist CP55940 for 30 mins and measured after 20 mins by Tango assay | Homo sapiens | 32 | ALA4364306 | cell-based format | Scientific Literature | |
8. | ALA4367896 | Binding | Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes at 10 uM incubated for 90 mins relative to control | Homo sapiens | 33 | ALA4364306 | cell-based format | Scientific Literature | |
9. | ALA4367897 | Binding | Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes at 10 uM incubated for 90 mins relative to control | Homo sapiens | 33 | ALA4364306 | cell-based format | Scientific Literature |