# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4404099 | Binding | Agonist activity at GST-tagged human FXR-LBD (193 to 472 residues) using biotinylated SRC-1 peptide as substrate incubated for 1 hrs by HTRF assay | Homo sapiens | 26 | ALA4402557 | single protein format | Scientific Literature | |
2. | ALA4404100 | Binding | Agonist activity at GST-tagged human FXR-LBD (193 to 472 residues) using biotinylated SRC-1 peptide as substrate incubated for 1 hrs by HTRF assay relative to GW4064 | Homo sapiens | 26 | ALA4402557 | single protein format | Scientific Literature | |
3. | ALA4404101 | Binding | Agonist activity at FXR transfected in human HEK293T cells o-expressing pGL3/hBSEP/luc incubated for 24 hrs by Steady-Glo reagent based luciferase reporter gene assay | Homo sapiens | 24 | ALA4402557 | cell-based format | Scientific Literature | |
4. | ALA4404102 | Binding | Agonist activity at FXR transfected in human HEK293T cells o-expressing pGL3/hBSEP/luc incubated for 24 hrs by Steady-Glo reagent based luciferase reporter gene assay relative to GW4064 | Homo sapiens | 24 | ALA4402557 | cell-based format | Scientific Literature |