1. ALA4324752 B Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins and measured every 2 secs for 120 secs by Fluo8-AM staining based FLIPR assay Homo sapiens 50 ALA4321858 cell-based format Scientific Literature 2. ALA4324753 A Transactivation of human PXR receptor expressed in HEPG2 or DPX2 cells co-expressing CYP3A4 promotor by One-Glo luciferase reporter gene assay Homo sapiens 50 ALA4321858 cell-based format Scientific Literature 3. ALA4324754 A Clearance in Han/Wistar rat hepatocytes assessed as extrapolated blood clearance at 1 uM and measured up to 90 mins by LC/MS/MS analysis Rattus norvegicus 29 ALA4321858 cell-based format Scientific Literature 4. ALA4725212 T Incucyte cell viability with HEK293T Homo sapiens 1,713 ALA4689842 cell-based format EUbOPEN Chemogenomic Library 5. ALA4725213 T Incucyte cell viability with human fibroblast Homo sapiens 1,718 ALA4689842 cell-based format EUbOPEN Chemogenomic Library 6. ALA4725214 T Incucyte cell viability with U2OS Homo sapiens 1,712 ALA4689842 cell-based format EUbOPEN Chemogenomic Library 7. ALA4879555 B KinomeScan assay: inhibition of AAK1 Homo sapiens 108 ALA4507330 single protein format Donated Chemical Probes - SGC Frankfurt 8. ALA4879556 B KinomeScan assay: inhibition of ABL1(E255K)-phosphorylated Homo sapiens 108 ALA4507330 single protein format Donated Chemical Probes - SGC Frankfurt 9. ALA4879557 B KinomeScan assay: inhibition of ABL1(F317I)-nonphosphorylated Homo sapiens 108 ALA4507330 single protein format Donated Chemical Probes - SGC Frankfurt 10. ALA4879558 B KinomeScan assay: inhibition of ABL1(F317I)-phosphorylated Homo sapiens 108 ALA4507330 single protein format Donated Chemical Probes - SGC Frankfurt 11. ALA4879559 B KinomeScan assay: inhibition of ABL1(F317L)-nonphosphorylated Homo sapiens 108 ALA4507330 single protein format Donated Chemical Probes - SGC Frankfurt 12. ALA4879560 B KinomeScan assay: inhibition of ABL1(F317L)-phosphorylated Homo sapiens 108 ALA4507330 single protein format Donated Chemical Probes - SGC Frankfurt 13. ALA4879561 B KinomeScan assay: inhibition of ABL1(H396P)-nonphosphorylated Homo sapiens 108 ALA4507330 single protein format Donated Chemical Probes - SGC Frankfurt 14. ALA4879562 B KinomeScan assay: inhibition of ABL1(H396P)-phosphorylated Homo sapiens 108 ALA4507330 single protein format Donated Chemical Probes - SGC Frankfurt 15. ALA4879563 B KinomeScan assay: inhibition of ABL1(M351T)-phosphorylated Homo sapiens 108 ALA4507330 single protein format Donated Chemical Probes - SGC Frankfurt 16. ALA4879564 B KinomeScan assay: inhibition of ABL1(Q252H)-nonphosphorylated Homo sapiens 108 ALA4507330 single protein format Donated Chemical Probes - SGC Frankfurt 17. ALA4879565 B KinomeScan assay: inhibition of ABL1(Q252H)-phosphorylated Homo sapiens 108 ALA4507330 single protein format Donated Chemical Probes - SGC Frankfurt 18. ALA4879566 B KinomeScan assay: inhibition of ABL1(T315I)-nonphosphorylated Homo sapiens 108 ALA4507330 single protein format Donated Chemical Probes - SGC Frankfurt 19. ALA4879567 B KinomeScan assay: inhibition of ABL1(T315I)-phosphorylated Homo sapiens 108 ALA4507330 single protein format Donated Chemical Probes - SGC Frankfurt 20. ALA4879568 B KinomeScan assay: inhibition of ABL1(Y253F)-phosphorylated Homo sapiens 108 ALA4507330 single protein format Donated Chemical Probes - SGC Frankfurt