# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4334826 | Binding | Inhibition of human immunoproteasome beta 5i subunit using Suc-LLVY-AMC as substrate preincubated for 30 mins followed by substrate addition and measured for 120 mins by fluorescence based assay | Homo sapiens | 12 | ALA4334435 | single protein format | Scientific Literature | |
2. | ALA4334829 | Binding | Inhibition of human immunoproteasome beta 2i subunit at 10 uM using Boc-LRR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay | Homo sapiens | 10 | ALA4334435 | single protein format | Scientific Literature | |
3. | ALA4334830 | Binding | Inhibition of human immunoproteasome beta 1i subunit at 10 uM using Ac-PAL-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay | Homo sapiens | 10 | ALA4334435 | single protein format | Scientific Literature | |
4. | ALA4334831 | ADME | Inhibition of human constitutive proteasome beta 5 subunit at 10 uM using Suc-LLVY-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay | Homo sapiens | 10 | ALA4334435 | single protein format | Scientific Literature | |
5. | ALA4334832 | ADME | Inhibition of human constitutive proteasome beta 2 subunit at 10 uM using Boc-LRR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay | Homo sapiens | 10 | ALA4334435 | single protein format | Scientific Literature | |
6. | ALA4334833 | ADME | Inhibition of human constitutive proteasome beta 1 subunit at 10 uM using Z-LLE-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay | Homo sapiens | 10 | ALA4334435 | single protein format | Scientific Literature | |
7. | ALA4334851 | Binding | Inhibition of human immunoproteasome beta 2i subunit using Boc-LRR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay | Homo sapiens | 10 | ALA4334435 | single protein format | Scientific Literature | |
8. | ALA4334852 | Binding | Inhibition of human immunoproteasome beta 1i subunit using Ac-PAL-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay | Homo sapiens | 10 | ALA4334435 | single protein format | Scientific Literature | |
9. | ALA4334853 | ADME | Inhibition of human constitutive proteasome beta 5 subunit using Suc-LLVY-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay | Homo sapiens | 10 | ALA4334435 | single protein format | Scientific Literature | |
10. | ALA4334854 | ADME | Inhibition of human constitutive proteasome beta 2 subunit using Boc-LRR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay | Homo sapiens | 10 | ALA4334435 | single protein format | Scientific Literature | |
11. | ALA4334855 | ADME | Inhibition of human constitutive proteasome beta 1 subunit using Z-LLE-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay | Homo sapiens | 10 | ALA4334435 | single protein format | Scientific Literature |