| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4429694 | B | Inhibition of human JAK1 at 1 uM using GEEPLYWSFPAKKK as substrate measured after 40 mins in presence of ATP by scintillation counting method | Homo sapiens | 48 | ALA4428074 | single protein format | Scientific Literature | |
| 2. | ALA4429696 | B | Inhibition of recombinant human C-terminal 6His-tagged JAK2 (808 to end amino acids) expressed in Sf21 cells at 1 uM measured after 1 hr in presence of ATP by TR-FRET assay | Homo sapiens | 48 | ALA4428074 | cell-based format | Scientific Literature | |
| 3. | ALA4429697 | B | Inhibition of recombinant human C-terminal 6His-tagged JAK2 (808 to end amino acids) expressed in Sf21 cells measured after 1 hr in presence of ATP by TR-FRET assay | Homo sapiens | 14 | ALA4428074 | cell-based format | Scientific Literature | |
| 4. | ALA4429698 | B | Inhibition of JAK3 (unknown origin) at 1 uM measured after 1 hr in presence of ATP by TR-FRET assay | Homo sapiens | 48 | ALA4428074 | single protein format | Scientific Literature | |
| 5. | ALA4429701 | B | Inhibition of JAK2 JH1/JH2 V617F mutant (unknown origin) at 100 nM measured after 1 hr in presence of ATP | Homo sapiens | 7 | ALA4428074 | single protein format | Scientific Literature | |
| 6. | ALA4429702 | F | Antiproliferative activity against HEL 92.1.7 cells assessed as viable cells at 10 uM measured after 3 days by WST-1 assay | Homo sapiens | 7 | ALA4428074 | cell-based format | Scientific Literature |
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