| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4414145 | B | Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assay relative to control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 2. | ALA4414146 | B | Inhibition of recombinant human catalytic GST-tagged ACVR1 expressed in baculovirus expression system assessed as reduction in enzyme activity at 5 uM in presence of ATP relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 3. | ALA4414147 | B | Inhibition of recombinant full length human GST-tagged CK1gamma1 expressed in baculovirus expression system assessed as reduction in enzyme activity at 5 uM in presence of ATP relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 4. | ALA4414148 | B | Selectivity ratio of IC50 for human GST-tagged CK2alpha H160A mutant to IC50 for human wild type GST-tagged CK2alpha | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 5. | ALA4414149 | B | Selectivity ratio of IC50 for human GST-tagged CK2alpha V73A mutant to IC50 for human wild type GST-tagged CK2alpha | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 6. | ALA4414150 | B | Selectivity ratio of IC50 for human GST-tagged CK2alpha L77A mutant to IC50 for human wild type GST-tagged CK2alpha | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 7. | ALA4414151 | B | Inhibition of recombinant human GST-tagged CK2alpha H160A mutant in presence of ATP by radiometric kinase assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA4414152 | B | Inhibition of recombinant full length human His-tagged GSK3beta expressed in baculovirus expression system assessed as reduction in enzyme activity at 5 uM in presence of ATP relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 9. | ALA4414153 | B | Inhibition of human PI3K assessed as reduction in enzyme activity at 5 uM in presence of ATP relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 10. | ALA4414154 | B | Inhibition of recombinant full length human His-tagged PIM1 expressed in baculovirus expression system assessed as reduction in enzyme activity at 5 uM in presence of ATP relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 11. | ALA4414155 | B | Inhibition of recombinant full length human His-tagged AURKB expressed in baculovirus expression system assessed as reduction in enzyme activity at 5 uM in presence of ATP relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 12. | ALA4414156 | B | Inhibition of human His-tagged ERBB2 expressed in baculovirus expression system assessed as reduction in enzyme activity at 5 uM in presence of ATP relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 13. | ALA4414157 | B | Inhibition of CK2alpha (unknown origin) assessed as reduction in enzyme activity at 5 uM in presence of ATP relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA4414158 | B | Inhibition of CK2 in human 786-0 cells assessed as decrease in alpha-catenin phosphorylation at Ser641 assuming basal level of non-responsive P-alpha-catenin of 50% of DMSO control after 24 hrs by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 15. | ALA4414159 | B | Inhibition of recombinant full length human GST-tagged CLK4 expressed in baculovirus expression system assessed as reduction in enzyme activity at 5 uM in presence of ATP relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 16. | ALA4414160 | B | Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assay | Homo sapiens | 23 | single protein format | Scientific Literature | ||
| 17. | ALA4414161 | B | Binding affinity to recombinant human GST-tagged CK2alpha after 120 secs by surface plasmon resonance analysis | Homo sapiens | 21 | single protein format | Scientific Literature | ||
| 18. | ALA4414162 | B | Inhibition of recombinant human GST-tagged CK2alpha at 10 uM in presence of ATP by radiometric kinase assay relative to control | Homo sapiens | 7 | single protein format | Scientific Literature | ||
| 19. | ALA4414163 | F | Growth inhibition of human 786-0 cells at 25 uM after 24 hrs by MTT assay relative to control | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 20. | ALA4414164 | B | Competitive inhibition of recombinant human GST-tagged CK2alpha by Lineweaver-Burk plot analysis | Homo sapiens | 1 | single protein format | Scientific Literature |
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