| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4310080 | Binding | Inhibition of BRD4 C-terminal bromodomain 2 (unknown origin) expressed in Escherichia coli Bl21(DE3) by alpha-screen assay | Homo sapiens | 4 | ALA4308848 | assay format | Scientific Literature | |
| 2. | ALA4310081 | Binding | Inhibition of BRD4 N-terminal bromodomain 1 (unknown origin) expressed in Escherichia coli Bl21(DE3) by alpha-screen assay | Homo sapiens | 4 | ALA4308848 | assay format | Scientific Literature | |
| 3. | ALA4310082 | Binding | Inhibition of BRD4 bromodomain 2 (unknown origin) expressed in Escherichia coli Bl21(DE3) by fluorescence anisotropy | Homo sapiens | 7 | ALA4308848 | assay format | Scientific Literature | |
| 4. | ALA4310083 | Binding | Inhibition of BRD4 bromodomain 1 (unknown origin) expressed in Escherichia coli Bl21(DE3) by fluorescence anisotropy | Homo sapiens | 6 | ALA4308848 | assay format | Scientific Literature | |
| 5. | ALA4310084 | Binding | Inhibition of human BRDT bromodomain 1 (unknown origin) expressed in Escherichia coli Bl21(DE3) by fluorescence anisotropy | Homo sapiens | 6 | ALA4308848 | assay format | Scientific Literature | |
| 6. | ALA4310087 | Binding | Inhibition of human BRDT bromodomain 2 (unknown origin) expressed in Escherichia coli Bl21(DE3) by fluorescence anisotropy | Homo sapiens | 6 | ALA4308848 | assay format | Scientific Literature | |
| 7. | ALA4310090 | Binding | Binding affinity to human BRDT bromodomain 1 (unknown origin) expressed in Escherichia coli Bl21(DE3) at 12.5 to 100 uM by protein-observed fluorine NMR method | Homo sapiens | 1 | ALA4308848 | assay format | Scientific Literature | |
| 8. | ALA4310091 | Binding | Inhibition of BRD3 N-terminal bromodomain 1 (unknown origin) expressed in Escherichia coli Bl21(DE3) by alpha-screen assay | Homo sapiens | 4 | ALA4308848 | assay format | Scientific Literature | |
| 9. | ALA4310092 | Binding | Inhibition of BRD3 C-terminal bromodomain 2 (unknown origin) expressed in Escherichia coli Bl21(DE3) by alpha-screen assay | Homo sapiens | 4 | ALA4308848 | assay format | Scientific Literature | |
| 10. | ALA4310093 | Binding | Inhibition of BRD2 N-terminal bromodomain 1 (unknown origin) expressed in Escherichia coli Bl21(DE3) by alpha-screen assay | Homo sapiens | 4 | ALA4308848 | assay format | Scientific Literature | |
| 11. | ALA4310094 | Binding | Inhibition of BRD2 C-terminal bromodomain 2 (unknown origin) expressed in Escherichia coli Bl21(DE3) by alpha-screen assay | Homo sapiens | 4 | ALA4308848 | assay format | Scientific Literature | |
| 12. | ALA4310095 | Binding | Inhibition of BRDT N-terminal bromodomain 1 (unknown origin) expressed in Escherichia coli Bl21(DE3) by alpha-screen assay | Homo sapiens | 4 | ALA4308848 | assay format | Scientific Literature | |
| 13. | ALA4310096 | Binding | Displacement of BI-BODIPY from BRD4 C-terminal bromodomain 2 (unknown origin) expressed in Escherichia coli Bl21(DE3) by fluorescence polarization assay | Homo sapiens | 4 | ALA4308848 | assay format | Scientific Literature | |
| 14. | ALA4310097 | Binding | Displacement of BI-BODIPY from BRDT C-terminal bromodomain 2 (unknown origin) expressed in Escherichia coli Bl21(DE3) by fluorescence polarization assay | Homo sapiens | 3 | ALA4308848 | assay format | Scientific Literature | |
| 15. | ALA4310098 | Binding | Binding affinity to BRD4 bromodomain 1 (unknown origin) expressed in Escherichia coli Bl21(DE3) by isothermal-titration calorimetry | Homo sapiens | 2 | ALA4308848 | assay format | Scientific Literature | |
| 16. | ALA4310099 | Binding | Selectivity ratio of IC50 for BRD2 C-terminal bromodomain 2 (unknown origin) expressed in Escherichia coli Bl21(DE3) to IC50 for BRD4 N-terminal bromodomain 1 (unknown origin) expressed in Escherichia coli Bl21(DE3) | Homo sapiens | 1 | ALA4308848 | assay format | Scientific Literature | |
| 17. | ALA4310100 | Binding | Selectivity ratio of IC50 for BRD3 C-terminal bromodomain 2 (unknown origin) expressed in Escherichia coli Bl21(DE3) to IC50 for BRD4 N-terminal bromodomain 1 (unknown origin) expressed in Escherichia coli Bl21(DE3) | Homo sapiens | 1 | ALA4308848 | assay format | Scientific Literature | |
| 18. | ALA4310101 | Binding | Displacement of Fl-JQ1 from BRD4 C-terminal bromodomain 2 H437D mutant (unknown origin) expressed in Escherichia coli Bl21(DE3) by fluorescence polarization assay | Homo sapiens | 2 | ALA4308848 | assay format | Scientific Literature | |
| 19. | ALA4310103 | Binding | Inhibition of human BRD4 bromodomain 1 expressed in HEK293 cells at 10 uM relative to control | Homo sapiens | 1 | ALA4308848 | cell-based format | Scientific Literature | |
| 20. | ALA4310104 | Binding | Inhibition of human BRDT bromodomain 1 expressed in HEK293 cells at 10 uM relative to control | Homo sapiens | 1 | ALA4308848 | cell-based format | Scientific Literature |
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