| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4360722 | B | Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysis | Rattus norvegicus | 26 | cell membrane format | Scientific Literature | ||
| 2. | ALA4360725 | B | Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysis | Rattus norvegicus | 17 | cell membrane format | Scientific Literature | ||
| 3. | ALA4360726 | B | Displacement of [3H]Ile5,6-deltorphin-2 from DOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysis | Rattus norvegicus | 17 | cell membrane format | Scientific Literature | ||
| 4. | ALA4360727 | B | Displacement of [3H]HS-665 from KOR in guinea pig brain membranes after 60 mins by liquid scintillation analysis | Cavia porcellus | 17 | cell membrane format | Scientific Literature | ||
| 5. | ALA4360728 | B | Selectivity ratio, ratio of Ki for displacement of [3H]Ile5,6-deltorphin-2 from DOR in Wistar rat brain membranes to Ki for displacement of [3H]DAMGO from MOR in Wistar rat brain membranes | Rattus norvegicus | 13 | cell membrane format | Scientific Literature | ||
| 6. | ALA4360729 | B | Selectivity ratio of Ki for displacement of [3H]HS-665 from KOR in guinea pig brain membranes to Ki for displacement of [3H]DAMGO from MOR in Wistar rat brain membranes | 12 | cell membrane format | Scientific Literature | |||
| 7. | ALA4360730 | B | Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysis | Rattus norvegicus | 17 | cell membrane format | Scientific Literature | ||
| 8. | ALA4360750 | B | Agonist activity at MOR/CB1R/CB2R receptor in Wistar rat brain membranes at 10 uM after 60 mins by [35S]-GTPgammaS binding assay relative to control | Rattus norvegicus | 17 | cell membrane format | Scientific Literature | ||
| 9. | ALA4360751 | F | Antagonist activity at MOR in Wistar rat brain membranes at 10 uM in presence of oxycodone after 60 mins by [35S]-GTPgammaS binding assay relative to control | Rattus norvegicus | 3 | cell membrane format | Scientific Literature | ||
| 10. | ALA4360752 | F | Antagonist activity at MOR in Wistar rat brain membranes at 10 uM in presence of Tyr-D-Ala-Gly-Phe-NH2 after 60 mins by [35S]-GTPgammaS binding assay relative to control | Rattus norvegicus | 3 | cell membrane format | Scientific Literature | ||
| 11. | ALA4360753 | F | Antagonist activity at CB1R/CB2R in Wistar rat brain membranes at 10 uM in presence of JWH-018 after 60 mins by [35S]-GTPgammaS binding assay relative to control | Rattus norvegicus | 4 | cell membrane format | Scientific Literature | ||
| 12. | ALA4360754 | B | Antagonist activity at MOR/CB1R/CB2R in Wistar rat brain membranes at 10 uM in presence of N-[6-[[2-[[(4R,4aS,7aR,12bS)-4a-hydroxy-9-methoxy-3-methyl-2,4,5,6,7a,13-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline-7-ylidene]amino]oxyacetyl]amino]hexyl]-6-[3-(naphthalene-1-carbonyl)indol-1-yl]hexanamide after 60 mins by [35S]-GTPgammaS binding assay relative to control | Rattus norvegicus | 2 | cell membrane format | Scientific Literature | ||
| 13. | ALA4360755 | B | Antagonist activity at MOR/CB1R/CB2R in Wistar rat brain membranes at 10 uM in presence of (S)-N-((2R,8S)-18-(3-(1-naphthoyl)-1H-indol-1-yl)-8-benzyl-3,6,9,12-tetraoxo-4,7,10,13-tetraazaoctadecan-2-yl)-2-amino-3-(4-hydroxyphenyl)propanamide after 60 mins by liquid scintillation analysis relative to control | Rattus norvegicus | 2 | cell membrane format | Scientific Literature |
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