#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA4411915	Binding	Displacement of [3H]-mibolerone from recombinant wild-type GST-tagged androgen receptor LBD (unknown origin) after 16 hrs by scintillation counting analysis	Homo sapiens	40	ALA4411271	single protein format	Scientific Literature
2.	ALA4411916	Binding	Antagonist activity at human androgen receptor expressed in HEK293 cells assessed as inhibition of R1881-induced receptor transactivation after 24 hrs by luciferase reporter gene assay	Homo sapiens	41	ALA4411271	cell-based format	Scientific Literature
3.	ALA4411917	Binding	Induction of full length androgen receptor degradation in human LNCaP cells at 1 uM after 24 hrs in presence of R1881 by Western blot analysis relative to control	Homo sapiens	41	ALA4411271	cell-based format	Scientific Literature
4.	ALA4411918	Binding	Induction of androgen receptor splice variant mutant degradation in human 22RV1 cells at 10 uM after 24 hrs in presence of R1881 by Western blot analysis relative to control	Homo sapiens	41	ALA4411271	cell-based format	Scientific Literature
5.	ALA4411919	Functional	Antiproliferative activity against human MR49F cells after 3 days followed by compound wash and measured after 6 days by SRB assay	Homo sapiens	35	ALA4411271	cell-based format	Scientific Literature
6.	ALA4411924	ADME	Half life in mouse liver microsomes at 50 uM in presence of cofactors for phase 1 and 2 metabolism	Mus musculus	20	ALA4411271	microsome format	Scientific Literature
7.	ALA4411925	ADME	Intrinsic clearance in mouse liver microsomes at 50 uM in presence of cofactors for phase 1 and 2 metabolism	Mus musculus	20	ALA4411271	microsome format	Scientific Literature
8.	ALA4411932	Functional	Antiproliferative activity against human MR49F cells after 3 days followed by compound wash and measured after 6 days by CellTiter-Glo assay	Homo sapiens	3	ALA4411271	cell-based format	Scientific Literature
9.	ALA4411939	Functional	In vivo antagonist activity at androgen receptor in C57B/L6 mouse assessed as induction of seminal vesicles atrophy at 40 mg/kg/day, po for 14 days by Hershberger assay	Mus musculus	9	ALA4411271	organism-based format	Scientific Literature
10.	ALA4411940	Functional	In vivo antagonist activity at androgen receptor in Sprague-Dawley rat assessed as induction of seminal vesicles atrophy at 40 mg/kg/day, po for 14 days by Hershberger assay	Rattus norvegicus	2	ALA4411271	organism-based format	Scientific Literature
11.	ALA4411941	Functional	In vivo antagonist activity at androgen receptor in po dosed Sprague-Dawley rat assessed as induction of seminal vesicles atrophy administered for 14 days by Hershberger assay	Rattus norvegicus	2	ALA4411271	organism-based format	Scientific Literature
12.	ALA4411942	Functional	In vivo antagonist activity at androgen receptor in po dosed Sprague-Dawley rat assessed as induction of prostate atrophy administered for 14 days by Hershberger assay	Rattus norvegicus	2	ALA4411271	organism-based format	Scientific Literature
13.	ALA4411943	Functional	In vivo antagonist activity at androgen receptor in Sprague-Dawley rat assessed as change in seminal vesicles weight at 40 mg/kg/day, po for 14 days by Hershberger assay relative to control	Rattus norvegicus	2	ALA4411271	organism-based format	Scientific Literature
14.	ALA4411944	Functional	In vivo antagonist activity at androgen receptor in Sprague-Dawley rat assessed as change in prostate weight at 40 mg/kg/day, po for 14 days by Hershberger assay relative to control	Rattus norvegicus	2	ALA4411271	organism-based format	Scientific Literature
15.	ALA4411949	Binding	Antagonist activity at rat GR expressed in COS cells assessed as reduction in receptor transactivation incubated for 24 hrs by luciferase reporter gene assay	Rattus norvegicus	4	ALA4411271	cell-based format	Scientific Literature
16.	ALA4411954	Binding	Induction of androgen receptor splice variant mutant degradation in human 22RV1 cells after 24 hrs in presence of R1881 by Western blot analysis relative to control	Homo sapiens	3	ALA4411271	cell-based format	Scientific Literature