| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4479308 | Binding | Antagonist activity at human P2X7 receptor | Homo sapiens | 4 | ALA4477234 | single protein format | Scientific Literature | |
| 2. | ALA4479309 | Binding | Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as inhibition of BzATP-induced EtBr uptake measured after 2 hrs by fluorescence analysis | Homo sapiens | 51 | ALA4477234 | cell-based format | Scientific Literature | |
| 3. | ALA4479310 | Binding | Antagonist activity at human P2X7 receptor in LPS/IFN-gamma-differentiated human THP-1 cells assessed as suppression of BzATP-stimulated IL-1beta release per-incubated for 30 mins before BzATP addition and measured after 30 mins by ELISA | Homo sapiens | 27 | ALA4477234 | cell-based format | Scientific Literature |
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