| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4373375 | Binding | Inhibition of recombinant human N-terminal His-tagged PDE10A2 expressed in HEK293 cells using cAMP as substrate measured after 60 mins | Homo sapiens | 23 | ALA4371089 | cell-based format | Scientific Literature | |
| 2. | ALA4373376 | ADME | Intrinsic clearance in human hepatic microsomes | Homo sapiens | 17 | ALA4371089 | microsome format | Scientific Literature | |
| 3. | ALA4373377 | ADME | Intrinsic clearance in rat hepatic microsomes | Rattus norvegicus | 17 | ALA4371089 | microsome format | Scientific Literature | |
| 4. | ALA4373378 | ADME | Apparent permeability in MDCK-MDR1 cells expressing human P-gp by transwell assay | Canis lupus familiaris | 21 | ALA4371089 | cell-based format | Scientific Literature | |
| 5. | ALA4373379 | ADME | Efflux ratio of apparent permeability from basolateral to apical over apical to basolateral side in MDCK-MDR1 cells expressing human P-gp | Canis lupus familiaris | 21 | ALA4371089 | cell-based format | Scientific Literature | |
| 6. | ALA4373380 | ADME | Inhibition of human PDE2A using cAMP as substrate measured after 60 mins | Homo sapiens | 11 | ALA4371089 | single protein format | Scientific Literature | |
| 7. | ALA4373381 | ADME | Inhibition of human GST-tagged PDE3A (484 to end residues) using cAMP as substrate measured after 60 mins | Homo sapiens | 14 | ALA4371089 | single protein format | Scientific Literature | |
| 8. | ALA4373382 | ADME | Inhibition of human full-length PDE4D2 expressed in Sf9 insect cells using cAMP as substrate measured after 60 mins | Homo sapiens | 16 | ALA4371089 | cell-based format | Scientific Literature |
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