#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA4323785	F	Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed by agonist solution addition after 60 mins by cell based TR-FRET assay	Homo sapiens	35	ALA4321836	cell-based format	Scientific Literature
2.	ALA4323786	A	Agonist activity at human luteinizing hormone receptor incubated for 60 mins by cell based TR-FRET assay	Homo sapiens	3	ALA4321836	cell-based format	Scientific Literature
3.	ALA4323787	F	Downregulation of human luteinizing hormone-induced COX-2 mRNA expression in cetrorelix-treated iv dosed female rat after 2 hrs by Taqman probe based RT-PCR analysis	Rattus norvegicus	1	ALA4321836	organism-based format	Scientific Literature
4.	ALA4323788	F	Reversal of human luteinizing hormone-induced suppression of aromatase mRNA expression in cetrorelix-treated iv dosed female rat after 2 hrs by Taqman probe based RT-PCR analysis	Rattus norvegicus	1	ALA4321836	organism-based format	Scientific Literature
5.	ALA4323789	F	Downregulation of human luteinizing hormone-induced RUNX1 mRNA expression in cetrorelix-treated iv dosed female rat after 2 hrs by Taqman probe based RT-PCR analysis	Rattus norvegicus	1	ALA4321836	organism-based format	Scientific Literature
6.	ALA4323790	F	Downregulation of human luteinizing hormone-induced Egr-1 mRNA expression in cetrorelix-treated iv dosed female rat after 2 hrs by Taqman probe based RT-PCR analysis	Rattus norvegicus	1	ALA4321836	organism-based format	Scientific Literature
7.	ALA4323791	B	Negative allosteric modulation of human luteinizing hormone receptor assessed as Emax for glycoprotein human luteinizing hormone-induced agonist activity at 0.84 nM to 17 uM preincubated for 20 mins followed by 100 times EC80 of agonist addition and measured after 60 mins by cell based TR-FRET assay relative to control	Homo sapiens	1	ALA4321836	cell-based format	Scientific Literature
8.	ALA4323792	A	Apparent permeability across apical to basolateral side in human Caco2 cells at 2 uM after 2 hrs by LC-MS/MS analysis	Homo sapiens	2	ALA4321836	cell-based format	Scientific Literature
9.	ALA4323793	B	Agonist activity at human A2B receptor expressed in HEK293 cells at 10 uM after 10 mins by HTRF assay relative to control	Homo sapiens	2	ALA4321836	cell-based format	Scientific Literature
10.	ALA4323794	F	Antagonist activity at human follicle stimulating hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed by agonist solution addition and measured after 120 mins by cell based TR-FRET assay	Homo sapiens	5	ALA4321836	cell-based format	Scientific Literature
11.	ALA4323796	F	Antagonist activity at rat luteinizing hormone receptor expressed in rat ovary granulosa GLHR15 cell suspension assessed as reduction in agonist-induced cAMP production preincubated for 30 mins followed by agonist solution addition after 30 mins by cell based TR-FRET assay	Rattus norvegicus	5	ALA4321836	cell-based format	Scientific Literature
12.	ALA4323797	F	Antagonist activity at human thyroid stimulating hormone receptor expressed in rat HTC133 cells assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed by agonist solution addition and measured after 60 mins by cell based TR-FRET assay	Homo sapiens	5	ALA4321836	cell-based format	Scientific Literature
13.	ALA4323799	P	Lipophilicity, logD of the compound at pH 7.5 by reversed-phase HPLC		32	ALA4321836	small-molecule physicochemical format	Scientific Literature
14.	ALA4323800	A	Clearance in human liver microsomes at 1 uM measured after 2 to 60 mins in presence of glucose-6-phosphate by LC-MS/MS analysis	Homo sapiens	30	ALA4321836	microsome format	Scientific Literature
15.	ALA4323801	A	Maximum oral bioavailability in human liver microsomes based well stirred liver model at 1 uM measured after 2 to 60 mins in presence of glucose-6-phosphate by LC-MS/MS analysis	Homo sapiens	30	ALA4321836	organism-based format	Scientific Literature
16.	ALA4323802	B	Antagonist activity at cynomolgus monkey luteinizing hormone receptor expressed in HEK293 cells assessed as reduction in agonist-induced cAMP production preincubated for 30 mins followed by agonist solution addition and measured after 30 mins by cell based TR-FRET assay	Macaca fascicularis	2	ALA4321836	cell-based format	Scientific Literature
17.	ALA4323803	A	Protein binding in human plasma assessed as unbound fraction	Homo sapiens	2	ALA4321836	cell-free format	Scientific Literature
18.	ALA4323804	B	Inhibition of human ERG expressed in HEK293 cells at holding potential -80 mV by whole-cell voltage-clamp method	Homo sapiens	2	ALA4321836	cell-based format	Scientific Literature
19.	ALA4323805	P	Aqueous solubility of the compound at pH 6.5 incubated for 24 hrs under shaking condition by HPLC-MS/MS analysis		2	ALA4321836	small-molecule physicochemical format	Scientific Literature
20.	ALA4323806	P	Chemical stability of the compound at pH 1 to 10 measured after 1 to 24 hrs by HPLC-UV method		2	ALA4321836	small-molecule physicochemical format	Scientific Literature