# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4386142 | Binding | Inhibition of His-tagged CDK2/Cyclin-E1 (unknown origin) expressed in baculovirus infected Sf9 insect cells using histone H1 as substrate measured in presence of [gamma-33P]ATP | Homo sapiens | 39 | ALA4385606 | cell-based format | Scientific Literature | |
2. | ALA4386143 | Functional | Antiproliferative activity against human HT cells measured after 72 hrs by calcein AM dye-based fluorescence assay | Homo sapiens | 39 | ALA4385606 | cell-based format | Scientific Literature | |
3. | ALA4386144 | Functional | Antiproliferative activity against human OCI-Ly2 cells measured after 72 hrs by calcein AM dye-based fluorescence assay | Homo sapiens | 39 | ALA4385606 | cell-based format | Scientific Literature | |
4. | ALA4386145 | Functional | Antiproliferative activity against human Mino cells measured after 72 hrs by calcein AM dye-based fluorescence assay | Homo sapiens | 39 | ALA4385606 | cell-based format | Scientific Literature | |
5. | ALA4386146 | Binding | Inhibition of His-tagged CDK1/Cyclin-B1 (unknown origin) expressed in baculovirus infected Sf9 insect cells using histone H1 as substrate measured in presence of [gamma-33P]ATP | Homo sapiens | 3 | ALA4385606 | cell-based format | Scientific Literature | |
6. | ALA4386147 | Binding | Inhibition of GST-tagged CDK2/Cyclin-A2 (unknown origin) expressed in Escherichia coli using histone H1 as substrate measured in presence of [gamma-33P]ATP | Homo sapiens | 3 | ALA4385606 | assay format | Scientific Literature | |
7. | ALA4386148 | Binding | Inhibition of recombinant human N-terminal GST-fused CDK4 (S4 to E303 residues)/cyclin D1 (Q4 to I295 residues) expressed in baculovirus infected Sf9 insect cells using RPPTLSPIPHIPR as substrate measured in presence of [gamma-33P]ATP | Homo sapiens | 3 | ALA4385606 | cell-based format | Scientific Literature | |
8. | ALA4386149 | Binding | Inhibition of recombinant human full-length N-terminal GST-His6 fused CDK5 (M1 to P292 residues)/N-terminal His6-tagged p25 (A104 to R307 residues) expressed in baculovirus infected Sf9 insect cells using histone H1 as substrate measured in presence of [gamma-33P]ATP | Homo sapiens | 3 | ALA4385606 | cell-based format | Scientific Literature | |
9. | ALA4386150 | Binding | Inhibition of recombinant human N-terminal GST-His6-fused CDK7 (M1 to F346 residues)/N-terminal His-tagged cyclin H (M1 to L323 residues)/N-terminal His6-tagged MAT1 (M1 to S306 residues) expressed in baculovirus infected Sf9 insect cells using (YSPTSPS)2KK as substrate measured in presence of [gamma-33P]ATP | Homo sapiens | 3 | ALA4385606 | cell-based format | Scientific Literature | |
10. | ALA4386151 | Binding | Inhibition of recombinant human N-terminal GST-His6-fused CDK9 (M1 to F372 residues)/N-terminal His6-tagged cyclin T1 (M1 to K726 residues) expressed in baculovirus infected Sf9 insect cells using (YSPTSPS)2KK as substrate measured in presence of [gamma-33P]ATP | Homo sapiens | 3 | ALA4385606 | cell-based format | Scientific Literature | |
11. | ALA4386152 | Binding | Inhibition of CK1delta (unknown origin) assessed as residual activity at 1 uM relative to control | Homo sapiens | 1 | ALA4385606 | single protein format | Scientific Literature | |
12. | ALA4386153 | Binding | Inhibition of CHK2 (unknown origin) assessed as residual activity at 1 uM relative to control | Homo sapiens | 1 | ALA4385606 | single protein format | Scientific Literature | |
13. | ALA4386154 | Binding | Inhibition of CK1delta (unknown origin) | Homo sapiens | 1 | ALA4385606 | single protein format | Scientific Literature | |
14. | ALA4386155 | Binding | Inhibition of CHK2 (unknown origin) | Homo sapiens | 1 | ALA4385606 | single protein format | Scientific Literature | |
15. | ALA4386156 | Functional | Antiproliferative activity against human RIVA cells assessed as growth inhibition measured after 72 hrs by calcein AM dye-based fluorescence assay | Homo sapiens | 2 | ALA4385606 | cell-based format | Scientific Literature | |
16. | ALA4386157 | Functional | Antiproliferative activity against human OCI-LY3 cells assessed as growth inhibition measured after 72 hrs by calcein AM dye-based fluorescence assay | Homo sapiens | 2 | ALA4385606 | cell-based format | Scientific Literature | |
17. | ALA4386158 | Functional | Antiproliferative activity against human U2932 cells assessed as growth inhibition measured after 72 hrs by calcein AM dye-based fluorescence assay | Homo sapiens | 2 | ALA4385606 | cell-based format | Scientific Literature | |
18. | ALA4386159 | Functional | Antiproliferative activity against human HBL1 cells assessed as growth inhibition measured after 72 hrs by calcein AM dye-based fluorescence assay | Homo sapiens | 2 | ALA4385606 | cell-based format | Scientific Literature | |
19. | ALA4386160 | Functional | Antiproliferative activity against human TMD8 cells assessed as growth inhibition measured after 72 hrs by calcein AM dye-based fluorescence assay | Homo sapiens | 2 | ALA4385606 | cell-based format | Scientific Literature | |
20. | ALA4386161 | Functional | Antiproliferative activity against human OCI-Ly2 cells assessed as growth inhibition measured after 72 hrs by calcein AM dye-based fluorescence assay | Homo sapiens | 2 | ALA4385606 | cell-based format | Scientific Literature |