#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA4400458	Binding	Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as substrate measured at 30 secs interval for 5 mins by FLINT assay	Homo sapiens	28	ALA4396973	cell-based format	Scientific Literature
2.	ALA4400459	ADME	Inhibition of human recombinant N-terminal His-tagged and enterokinase cleavage site-fused KLK1 (19 to 262 residues) expressed in baculovirus infected Sf9 insect cells using R110 labelled GSK3162232A as substrate measured at 30 secs interval for 5 mins by FLINT assay	Homo sapiens	28	ALA4396973	cell-based format	Scientific Literature
3.	ALA4400460	Physicochemical	Dissociation constant, borocycle pKa of the compound		10	ALA4396973	small-molecule physicochemical format	Scientific Literature
4.	ALA4400461	Binding	Inhibition of human recombinant N-terminal His-tagged and enterokinase cleavage site-fused KLK1 (19 to 262 residues) expressed in baculovirus infected Sf9 insect cells at 10 uM using R110 labelled GSK3162232A as substrate measured at 30 secs interval for 5 mins by FLINT assay relative to control	Homo sapiens	7	ALA4396973	cell-based format	Scientific Literature
5.	ALA4400462	ADME	Inhibition of recombinant human C-terminal 10-His-tagged factor Xa (L24 to K488 residues) expressed in baculovirus infected Sf21 insect cells using Mca-RPKPVE-Nval-WRK(Dnp)-NH2 as substrate incubated for 40 mins by FLINT assay	Homo sapiens	15	ALA4396973	cell-based format	Scientific Literature
6.	ALA4400463	Binding	Inhibition of human C-terminal 6-His-tagged KLKB1 (G20-A638 residues) expressed in mouse NS0 cells using PFR-AMC as substrate incubated for 40 mins by FLINT assay	Homo sapiens	15	ALA4396973	cell-based format	Scientific Literature
7.	ALA4400464	Binding	Inhibition of recombinant human C-terminal 10-His-tagged KLK7 (Glu23 to His252 residues) expressed in mouse NS0 cells using 5-FAM-E-A-L-Y-L-V-S-G-C(5-TAMRA) as substrate incubated for 40 mins by FLINT assay	Homo sapiens	15	ALA4396973	cell-based format	Scientific Literature
8.	ALA4400465	Binding	Inhibition of recombinant human C-terminal 10-His-tagged KLK8 (Gln29 to Gly260 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate incubated for 40 mins by FLINT assay	Homo sapiens	15	ALA4396973	cell-based format	Scientific Literature
9.	ALA4400466	Binding	Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate incubated for 40 mins by FLINT assay	Homo sapiens	15	ALA4396973	cell-based format	Scientific Literature
10.	ALA4400467	ADME	Inhibition of recombinant human N-terminal Met and 6-His-tagged matriptase (G596 to V855 residues) expressed in Escherichia coli using Boc-QAR-AMC as substrate incubated for 40 mins by FLINT assay	Homo sapiens	15	ALA4396973	assay format	Scientific Literature
11.	ALA4400468	ADME	Inhibition of human recombinant C-terminal 10-His-tagged thrombin (M1 to E622 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate incubated for 40 mins by FLINT assay	Homo sapiens	15	ALA4396973	cell-based format	Scientific Literature
12.	ALA4400469	ADME	Inhibition of human neutrophil elastase using MeOSuc-AAPV-AMC as substrate incubated for 40 mins by FLINT assay	Homo sapiens	15	ALA4396973	single protein format	Scientific Literature
13.	ALA4400470	ADME	Inhibition of recombinant human C-terminal 10-His-tagged urokinase (M1 to L431 residues) expressed in mouse NS0 cells using Z-GGR-AMC as substrate incubated for 40 mins by FLINT assay	Homo sapiens	15	ALA4396973	cell-based format	Scientific Literature
14.	ALA4400476	Binding	Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as substrate measured at 30 secs interval for 5 mins using 1 x 10'10M enzyme by FLINT assay	Homo sapiens	15	ALA4396973	cell-based format	Scientific Literature
15.	ALA4400477	Binding	Selectivity ratio of IC50 for human C-terminal 6-His-tagged KLKB1 (G20 to A638 residues) expressed in mouse NS0 cells to IC50 for human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells	Homo sapiens	15	ALA4396973	cell-based format	Scientific Literature