| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4312523 | A | Drug metabolism in iv or po dosed dog assessed as PT2385 formation | Canis lupus familiaris | 1 | ALA4311943 | organism-based format | Scientific Literature | |
| 2. | ALA4312530 | A | Drug level in human hepatocytes treated with PT2385 assessed as metabolite formation by HPLC-UV analysis | Homo sapiens | 1 | ALA4311943 | cell-based format | Scientific Literature | |
| 3. | ALA4312553 | A | Substrate activity at BCRP (unknown origin) expressed in MDCK2 cells assessed as efflux ratio of permeability at up to 300 uM | Homo sapiens | 2 | ALA4311943 | cell-based format | Scientific Literature | |
| 4. | ALA4312554 | A | Substrate activity at P-gp (unknown origin) expressed in MDCK2 cells assessed as efflux ratio of permeability at up to 300 uM | Homo sapiens | 2 | ALA4311943 | cell-based format | Scientific Literature | |
| 5. | ALA4312556 | A | Ratio of compound effect for substrate activity at human MRP2 expressed in Sf9 membrane vesicles assessed as protein-mediated drug uptake in presence of ATP to compound effect for substrate activity at human MRP2 expressed in Sf9 membrane vesicles assessed as protein-mediated drug uptake in absence of ATP | Homo sapiens | 1 | ALA4311943 | cell membrane format | Scientific Literature | |
| 6. | ALA4312557 | A | Substrate activity at human MRP2 expressed in Sf9 membrane vesicles assessed as Vmax per mg protein | Homo sapiens | 1 | ALA4311943 | cell-based format | Scientific Literature | |
| 7. | ALA4312558 | A | Substrate activity at human MRP2 expressed in Sf9 membrane vesicles assessed as Km | Homo sapiens | 1 | ALA4311943 | cell-based format | Scientific Literature | |
| 8. | ALA4312559 | A | Substrate activity at human MRP2 expressed in Sf9 membrane vesicles assessed as protein-mediated drug uptake in presence of MRP2 inhibitor-benzbromarone by LC-MS/MS analysis | Homo sapiens | 1 | ALA4311943 | cell-based format | Scientific Literature | |
| 9. | ALA4312560 | A | Drug metabolism assessed as Escherichia coli beta-glucuronidase-mediated PT2385 formation after 30 mins by LC-MS/MS analysis | Escherichia coli | 1 | ALA4311943 | single protein format | Scientific Literature |
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