| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4306826 | B | Inverse agonist activity at RORC2 in human Th17 cells assessed as inhibition of IL-17A secretion incubated for 4 days by HTRF assay | Homo sapiens | 29 | ALA4304769 | cell-based format | Scientific Literature | |
| 2. | ALA4306827 | B | Inverse agonist activity at RORC2 in human Th17 cells assessed as inhibition of IL-17A secretion incubated for 4 days by HTRF assay relative to control | Homo sapiens | 28 | ALA4304769 | cell-based format | Scientific Literature | |
| 3. | ALA4306828 | P | 1-Octanol/PBS buffer distribution coefficient, log D of the compound at pH 7.4 | 28 | ALA4304769 | small-molecule physicochemical format | Scientific Literature | ||
| 4. | ALA4306829 | P | Thermodynamic solubility of the compound in aqueous phosphate buffer at pH 7.4 measured after 24 hrs by UPLC-MS/MS-based shake-flask method | 28 | ALA4304769 | small-molecule physicochemical format | Scientific Literature | ||
| 5. | ALA4306842 | B | Agonist activity at LXR alpha (unknown origin) up to 10 uM by reporter gene assay | Homo sapiens | 1 | ALA4304769 | single protein format | Scientific Literature | |
| 6. | ALA4306843 | B | Agonist activity at LXR beta (unknown origin) up to 10 uM by reporter gene assay | Homo sapiens | 1 | ALA4304769 | single protein format | Scientific Literature | |
| 7. | ALA4306848 | B | Agonist activity at RORalpha (unknown origin) | Homo sapiens | 1 | ALA4304769 | single protein format | Scientific Literature | |
| 8. | ALA4306849 | B | Agonist activity at RORbeta (unknown origin) | Homo sapiens | 2 | ALA4304769 | single protein format | Scientific Literature | |
| 9. | ALA4306853 | B | Inverse agonist activity at human biotinylated HN-Avi-MBPS-TCS-RORC2 (258 to 518 residues) assessed as recruitment of SRC-1-derived coactivator peptide measured after 15 mins by FRET assay relative to control | Homo sapiens | 26 | ALA4304769 | single protein format | Scientific Literature | |
| 10. | ALA4306854 | B | Inverse agonist activity at human biotinylated HN-Avi-MBPS-TCS-RORC2 (258 to 518 residues) assessed as recruitment of SRC-1-derived coactivator measured after 15 mins by FRET assay | Homo sapiens | 28 | ALA4304769 | single protein format | Scientific Literature | |
| 11. | ALA4306855 | B | Agonist activity at RAR alpha (unknown origin) | Homo sapiens | 2 | ALA4304769 | single protein format | Scientific Literature | |
| 12. | ALA4306856 | B | Agonist activity at RAR beta (unknown origin) | Homo sapiens | 2 | ALA4304769 | single protein format | Scientific Literature | |
| 13. | ALA4306857 | B | Agonist activity at RAR gamma (unknown origin) | Homo sapiens | 2 | ALA4304769 | single protein format | Scientific Literature |
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