# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4479676 | B | Inhibition of full-length recombinant human GST-tagged MARK3 expressed in baculovirus expression system using biotinylated-Cdc25C peptide substrate measured after 2 hrs by HTRF assay | Homo sapiens | 27 | ALA4477252 | assay format | Scientific Literature | |
2. | ALA4479681 | A | Substrate activity at human MDR1 expressed in LLC-PK1 cells assessed as efflux ratio of permeability across basolateral to apical over apical to basolateral side at 5 uM | Homo sapiens | 7 | ALA4477252 | cell-based format | Scientific Literature | |
3. | ALA4479683 | A | Apparent permeability from basolateral to apical side over apical to basolateral side in pig LLC-PK1 cells expressing MDR1 (unknown origin) at 5 uM measured after 3 hrs | Sus scrofa | 4 | ALA4477252 | cell-based format | Scientific Literature | |
4. | ALA4479684 | P | Solubility of the compound at pH 7 | 15 | ALA4477252 | small-molecule physicochemical format | Scientific Literature |