| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4315162 | B | Inhibition of human SUV39H2 at 100 uM using histone H3 as substrate incubated for 1 hr in presence of [3H]-SAM by filter binding method relative to control | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature | |
| 2. | ALA4315163 | B | Inhibition of human SUV39H1 at 100 uM using histone H3 as substrate incubated for 1 hr in presence of [3H]-SAM by filter binding method relative to control | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature | |
| 3. | ALA4315164 | B | Inhibition of human SET7/9 at 100 uM using core histone as substrate incubated for 1 hr in presence of [3H]-SAM by filter binding method relative to control | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature | |
| 4. | ALA4315165 | B | Inhibition of human PRMT1 at 100 uM using histone H4 as substrate incubated for 1 hr in presence of [3H]-SAM by filter binding method relative to control | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature | |
| 5. | ALA4315166 | B | Inhibition of human MLL1 complex at 100 uM using core histone as substrate incubated for 1 hr in presence of [3H]-SAM by filter binding method relative to control | Homo sapiens | 1 | ALA4311997 | assay format | Scientific Literature | |
| 6. | ALA4315167 | B | Inhibition of human G9a at 100 uM using core histone H3 (1 to 21 residues) as substrate incubated for 1 hr in presence of [3H]-SAM by filter binding method relative to control | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature | |
| 7. | ALA4315168 | B | Inhibition of human EZH2 complex at 100 uM using core histone as substrate incubated for 1 hr in presence of [3H]-SAM by filter binding method relative to control | Homo sapiens | 1 | ALA4311997 | assay format | Scientific Literature | |
| 8. | ALA4315169 | B | Inhibition of human DOT1L at 100 uM using oligo nucleosomes as substrate incubated for 1 hr in presence of [3H]-SAM by filter binding method relative to control | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature | |
| 9. | ALA4315170 | B | Inhibition of human DNMT3a using lambda DNA as substrate incubated for 1 hr in presence of [3H]-SAM by filter binding method | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature | |
| 10. | ALA4315171 | B | Inhibition of human DNMT1 using Poly(dI-dC) as substrate incubated for 1 hr in presence of [3H]-SAM by filter binding method | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature | |
| 11. | ALA4315172 | B | Selectivity ratio of IC50 for human HDAC8 to IC50 for human HDAC6 | Homo sapiens | 1 | ALA4311997 | assay format | Scientific Literature | |
| 12. | ALA4315173 | B | Selectivity ratio of IC50 for human HDAC2 to IC50 for human HDAC6 | Homo sapiens | 1 | ALA4311997 | assay format | Scientific Literature | |
| 13. | ALA4315174 | B | Selectivity ratio of IC50 for human HDAC3 to IC50 for human HDAC6 | Homo sapiens | 1 | ALA4311997 | assay format | Scientific Literature | |
| 14. | ALA4315175 | B | Inhibition of human HDAC9 at 10 uM using Acetyl-Lys (trifluoroacetyl)-AMC) as substrate incubated for 2 hrs by fluorescence assay relative to control | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature | |
| 15. | ALA4315176 | B | Inhibition of human HDAC8 using Arg-His-Lys (Ac)-Lys (Ac) as substrate incubated for 2 hrs by fluorescence assay | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature | |
| 16. | ALA4315177 | B | Inhibition of human HDAC7 at 10 uM using Acetyl-Lys (trifluoroacetyl)-AMC) as substrate incubated for 2 hrs by fluorescence assay | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature | |
| 17. | ALA4315178 | B | Inhibition of human HDAC5 at 10 uM using Acetyl-Lys (trifluoroacetyl)-AMC) as substrate incubated for 2 hrs by fluorescence assay relative to control | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature | |
| 18. | ALA4315179 | B | Inhibition of human HDAC4 at 10 uM using Acetyl-Lys (trifluoroacetyl)-AMC) as substrate incubated for 2 hrs by fluorescence assay relative to control | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature | |
| 19. | ALA4315180 | B | Inhibition of human HDAC3 using Arg-His-Lys-Lys (Ac) as substrate incubated for 2 hrs by fluorescence assay | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature | |
| 20. | ALA4315182 | B | Inhibition of human HDAC2 using Arg-His-Lys-Lys (Ac) as substrate incubated for 2 hrs by fluorescence assay | Homo sapiens | 1 | ALA4311997 | single protein format | Scientific Literature |
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