| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4389076 | A | Clearance in human liver microsomes relative to hepatic blood flow | Homo sapiens | 2 | ALA4387741 | microsome format | Scientific Literature | |
| 2. | ALA4389078 | B | Reversible inhibition of recombinant full-length N-terminal 6-His-tagged human BTK expressed in baculovirus infected Sf21 insect cells using fluorescent-labeled polyGAT peptide as substrate incubated for 30 mins by TR-FRET assay | Homo sapiens | 33 | ALA4387741 | cell-based format | Scientific Literature | |
| 3. | ALA4389079 | B | Inhibition of human wild-type AAK1 (G25 to L333 residues) expressed in bacterial expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 4. | ALA4389080 | B | Inhibition of human phosphorylated ABL1 E255K mutant (S229 to K512 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 5. | ALA4389081 | B | Inhibition of human non-phosphorylated ABL1 F317I mutant (S229 to K512 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 6. | ALA4389082 | B | Inhibition of human phosphorylated ABL1 F317I mutant (S229 to K512 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 7. | ALA4389083 | B | Inhibition of human non-phosphorylated ABL1 F317L mutant (S229 to K512 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 8. | ALA4389084 | B | Inhibition of human phosphorylated ABL1 F317L mutant (S229 to K512 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 9. | ALA4389085 | B | Inhibition of human non-phosphorylated ABL1 H396P mutant (S229 to K512 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 10. | ALA4389086 | B | Inhibition of human phosphorylated ABL1 H396P mutant (S229 to K512 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 11. | ALA4389087 | B | Inhibition of human phosphorylated ABL1 M351T mutant (S229 to K512 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 12. | ALA4389088 | B | Inhibition of human non-phosphorylated ABL1 Q252H mutant (S229 to K512 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 13. | ALA4389089 | B | Inhibition of human phosphorylated ABL1 Q252H mutant expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 14. | ALA4389090 | B | Inhibition of human non-phosphorylated ABL1 T315I mutant (S229 to K512 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 15. | ALA4389091 | B | Inhibition of human phosphorylated ABL1 T315I mutant (S229 to K512 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 16. | ALA4389092 | B | Inhibition of human phosphorylated ABL1 Y253F mutant (S229 to K512 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 17. | ALA4389093 | B | Inhibition of wild-type human non-phosphorylated ABL1 (S229 to K512 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 18. | ALA4389094 | B | Inhibition of wild-type human phosphorylated ABL1 (S229 to K512 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 19. | ALA4389095 | B | Inhibition of wild-type human ABL2 (A248 to G542 residues) expressed in bacterial expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature | |
| 20. | ALA4389096 | B | Inhibition of wild-type human ACVR1 (C188 to C509 residues) expressed in bacterial expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4387741 | assay format | Scientific Literature |
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