#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA4477863	Functional	Antiproliferative activity against human 22Rv1 cells after 96 hrs by propidium iodide staining based fluorescence 2D monolayer assay	Homo sapiens	111	ALA4477199	cell-based format	Scientific Literature
2.	ALA4477864	Functional	Antiproliferative activity against human DU145 cells after 96 hrs by propidium iodide staining based fluorescence 2D monolayer assay	Homo sapiens	111	ALA4477199	cell-based format	Scientific Literature
3.	ALA4477865	Functional	Antiproliferative activity against human LNCAP cells after 96 hrs by propidium iodide staining based fluorescence 2D monolayer assay	Homo sapiens	111	ALA4477199	cell-based format	Scientific Literature
4.	ALA4477866	Functional	Antiproliferative activity against human VCaP cells after 96 hrs by propidium iodide staining based fluorescence 2D monolayer assay	Homo sapiens	111	ALA4477199	cell-based format	Scientific Literature
5.	ALA4477867	Physicochemical	Solubility in RPMI1640 culture medium at <30 uM incubated for 4 days by microscopic analysis		109	ALA4477199	small-molecule physicochemical format	Scientific Literature
6.	ALA4477868	Physicochemical	Solubility in 100% DMSO at 33 mM at -20 degC		109	ALA4477199	small-molecule physicochemical format	Scientific Literature
7.	ALA4477882	Binding	Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition of R1881-induced receptor activation at 10 uM preincubated for 30 mins followed by R1881 addition measured after 16 to 24 hrs by betalactamase reporter gene assay relative to control	Rattus norvegicus	23	ALA4477199	cell-based format	Scientific Literature
8.	ALA4477884	Binding	Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition of R1881-induced receptor activation preincubated for 30 mins followed by R1881 addition measured after 16 to 24 hrs by betalactamase reporter gene assay	Rattus norvegicus	26	ALA4477199	cell-based format	Scientific Literature
9.	ALA4477885	Binding	Agonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as receptor activation at 10 uM incubated for 16 to 24 hrs by betalactamase reporter gene assay relative to control	Rattus norvegicus	14	ALA4477199	cell-based format	Scientific Literature
10.	ALA4477886	ADME	Intrinsic clearance in human liver microsomes assessed per mg protein at 3 uM preincubated with compound followed by NADPH addition measured after 5 to 45 mins by LC-MS/MS analysis	Homo sapiens	10	ALA4477199	microsome format	Scientific Literature
11.	ALA4477888	ADME	Half life in human liver microsomes at 3 uM preincubated with compound followed by NADPH addition by LC-MS/MS analysis	Homo sapiens	10	ALA4477199	microsome format	Scientific Literature
12.	ALA4477889	ADME	Apparent permeability from apical to basolateral side in human Caco2 cells at 10 uM incubated for 120 mins by LC-MS/MS analysis	Homo sapiens	14	ALA4477199	cell-based format	Scientific Literature
13.	ALA4477890	ADME	Apparent permeability from basolateral to apical side in human Caco2 cells at 10 uM incubated for 120 mins by LC-MS/MS analysis	Homo sapiens	14	ALA4477199	cell-based format	Scientific Literature
14.	ALA4477891	ADME	Efflux ratio of apparent permeability from basolateral to apical side over apical to basolateral side in human Caco2 cells at 10 uM incubated for 120 mins by LC-MS/MS analysis	Homo sapiens	14	ALA4477199	cell-based format	Scientific Literature
15.	ALA4477892	Functional	Cytotoxicity against human HepG2 cells assessed as reduction in cell viability after 72 hrs by MTT assay	Homo sapiens	13	ALA4477199	cell-based format	Scientific Literature
16.	ALA4477898	Binding	Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition of R1881-induced receptor activation at 3160 nM preincubated for 30 mins followed by R1881 addition measured after 16 to 24 hrs by betalactamase reporter gene assay relative to control	Rattus norvegicus	5	ALA4477199	cell-based format	Scientific Literature
17.	ALA4477899	Binding	Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition of R1881-induced receptor activation at 1000 nM preincubated for 30 mins followed by R1881 addition measured after 16 to 24 hrs by betalactamase reporter gene assay relative to control	Rattus norvegicus	5	ALA4477199	cell-based format	Scientific Literature
18.	ALA4477900	Binding	Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition of R1881-induced receptor activation at 316 nM preincubated for 30 mins followed by R1881 addition measured after 16 to 24 hrs by betalactamase reporter gene assay relative to control	Rattus norvegicus	5	ALA4477199	cell-based format	Scientific Literature
19.	ALA4477901	Binding	Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition of R1881-induced receptor activation at 100 nM preincubated for 30 mins followed by R1881 addition measured after 16 to 24 hrs by betalactamase reporter gene assay relative to control	Rattus norvegicus	5	ALA4477199	cell-based format	Scientific Literature
20.	ALA4477902	Binding	Antagonist activity at rat androgen receptor fused with DNA-binding domain of GAL4 expressed in AR-UAS-bla GripTite 293 cells assessed as inhibition of R1881-induced receptor activation at 31.6 nM preincubated for 30 mins followed by R1881 addition measured after 16 to 24 hrs by betalactamase reporter gene assay relative to control	Rattus norvegicus	5	ALA4477199	cell-based format	Scientific Literature