| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4341825 | Binding | Antagonist activity at GST-tagged FXR LBD (unknown origin) assessed as inhibition of GW4064-induced fluorecein-labeled SRC2-2 coactivator recruitment by Lanthascreen TR-FRET assay | Homo sapiens | 21 | ALA4340545 | single protein format | Scientific Literature | |
| 2. | ALA4341826 | Binding | Antagonist activity at human FXR expressed in Huh7 cells assessed as inhibition of CDCA-induced FXR response element driven luciferase activity after 24 hrs | Homo sapiens | 21 | ALA4340545 | cell-based format | Scientific Literature | |
| 3. | ALA4341827 | ADME | Cytotoxicity against human HuH7 cells assessed as reduction in cell viability incubated for 24 hrs by MTT assay | Homo sapiens | 20 | ALA4340545 | cell-based format | Scientific Literature |
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