# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4411099 | B | Inhibition of human GRK5 using tubulin as substrate measured after 0 mins by [gamma-32P]-ATP assay | Homo sapiens | 7 | ALA4406919 | single protein format | Scientific Literature | |
2. | ALA4411102 | B | Inhibition of human GRK5 using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assay | Homo sapiens | 12 | ALA4406919 | single protein format | Scientific Literature | |
3. | ALA4411104 | B | Inhibition of bovine GRK2 using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assay | Bos taurus | 16 | ALA4406919 | single protein format | Scientific Literature | |
4. | ALA4411105 | B | Inhibition of bovine GRK6 using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assay | Bos taurus | 12 | ALA4406919 | assay format | Scientific Literature | |
5. | ALA4411106 | B | Inhibition of bovine GRK5 C474S mutant using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assay | Bos taurus | 5 | ALA4406919 | single protein format | Scientific Literature | |
6. | ALA4411108 | B | Selectivity index, ratio of IC50 for bovine GRK2 to IC50 for human GRK5 | 16 | ALA4406919 | assay format | Scientific Literature | ||
7. | ALA4411109 | B | Covalent inhibition of human GRK5 assessed as adduct appearance incubated for 3 hrs by intact protein mass spectroscopy | Homo sapiens | 11 | ALA4406919 | single protein format | Scientific Literature | |
8. | ALA4411110 | B | Covalent binding affinity to human GRK5 assessed as covalent bond formation with Cys474 by intact protein mass spectrometry | Homo sapiens | 1 | ALA4406919 | single protein format | Scientific Literature | |
9. | ALA4411111 | B | Covalent binding affinity to bovine GRK5 C474S mutant assessed as covalent bond formation with Cys474 by intact protein mass spectrometry | Bos taurus | 1 | ALA4406919 | single protein format | Scientific Literature | |
10. | ALA4411112 | B | Inhibition of human GRK5 using tubulin as substrate measured after 100 mins by [gamma-32P]-ATP assay | Homo sapiens | 1 | ALA4406919 | single protein format | Scientific Literature |