| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA640714 | A | Plasma half life in rat serum | Rattus norvegicus | 20 | organism-based format | Scientific Literature | ||
| 2. | ALA687141 | F | Relative potency expressed in percent to that of neurotensin was measured using guinea pig atria | 25 | assay format | Scientific Literature | |||
| 3. | ALA693866 | F | Compound was tested in vitro to mobilize calcium from HT-29 cells | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 4. | ALA720040 | F | Analgesic activity was evaluated in the acetic acid induced stretching paradigm after subcutaneous administration | Mus musculus | 3 | organism-based format | Scientific Literature | ||
| 5. | ALA721107 | F | Compound was tested in vivo for its ability to inhibit spontaneous locomotor activity of mice; intraperitoneal administration | Mus musculus | 4 | organism-based format | Scientific Literature | ||
| 6. | ALA731158 | F | Antinociceptive activity using the mouse phenylquinone writhing assay with i.c.v. administration | Mus musculus | 23 | organism-based format | Scientific Literature | ||
| 7. | ALA754783 | B | Binding affinity for Neurotensin Receptor | Mus musculus | 13 | single protein format | Scientific Literature | ||
| 8. | ALA754794 | B | Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum) | 17 | tissue-based format | Scientific Literature | |||
| 9. | ALA754795 | B | In vitro affinity for the neurotensin receptor on mouse brain membranes. | 23 | tissue-based format | Scientific Literature | |||
| 10. | ALA754342 | B | Tested for change in binding affinity in neonatal mouse whole brain (minus cerebellum) | 1 | tissue-based format | Scientific Literature | |||
| 11. | ALA754345 | B | IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracer | Rattus norvegicus | 7 | assay format | Scientific Literature | ||
| 12. | ALA754352 | B | Relative potency at neurotensin receptor compared to neurotensin (NT8-13) | Rattus norvegicus | 9 | single protein format | Scientific Literature | ||
| 13. | ALA754353 | B | Evaluated for binding affinity by inhibiting binding of [125I]-Tyr(3)-NT to human Neurotensin receptor 1 | 21 | single protein format | Scientific Literature | |||
| 14. | ALA754354 | B | Ability to compete with [125I]-Tyr(3)NT (0.15 nM) for human Neurotensin receptor 1 | 21 | single protein format | Scientific Literature | |||
| 15. | ALA754355 | B | Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2 | 21 | single protein format | Scientific Literature | |||
| 16. | ALA754356 | B | Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 3 | 21 | single protein format | Scientific Literature | |||
| 17. | ALA799610 | F | Relative potency expressed in percent to that of neurotensin was measured using rat stomach strips assay | 25 | tissue-based format | Scientific Literature | |||
| 18. | ALA801010 | F | Relative potency expressed in percent to that of neurotensin was measured using perfused rat heart assay | 25 | assay format | Scientific Literature | |||
| 19. | ALA829237 | B | In vitro inhibition of [3H]-NT binding to human striatal Neurotensin receptor 1 | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 20. | ALA840036 | B | In vitro inhibition of [3H]NT binding to porcine striatal Neurotensin receptor 1 | Sus scrofa | 6 | single protein format | Scientific Literature |
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