| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4338950 | B | Inhibition of recombinant N-terminal FLAG/His-tagged SMYD3 (unknown origin) expressed in baculovirus infected insect cells using 3H-SAM as substrate assessed as 3H-MEKK2 methylation incubated for 40 mins by scintillation proximity assay | Homo sapiens | 49 | cell-based format | Scientific Literature | ||
| 2. | ALA4338951 | B | Inhibition of recombinant SMYD3 (unknown origin) transfected in human HEK293 cells assessed as reduction in MEKK2 methylation incubated for 24 hrs by cellular mechanistic assay | Homo sapiens | 49 | cell-based format | Scientific Literature | ||
| 3. | ALA4338952 | P | Solubility of compound by CLND method | 47 | small-molecule physicochemical format | Scientific Literature | |||
| 4. | ALA4338953 | A | Permeability of compound | 44 | assay format | Scientific Literature | |||
| 5. | ALA4338964 | A | AUC in Sprague-Dawley rat at 2 mg/kg, po | Rattus norvegicus | 8 | organism-based format | Scientific Literature | ||
| 6. | ALA4338965 | A | Oral bioavailability in Sprague-Dawley rat at 2 mg/kg | Rattus norvegicus | 7 | organism-based format | Scientific Literature | ||
| 7. | ALA4338966 | A | Clearance in Sprague-Dawley rat at 1 mg/kg, iv or 2 mg/kg, po | Rattus norvegicus | 4 | organism-based format | Scientific Literature | ||
| 8. | ALA4338967 | A | Volume of distribution in Sprague-Dawley rat at 1 mg/kg, iv or 2 mg/kg, po | Rattus norvegicus | 4 | organism-based format | Scientific Literature | ||
| 9. | ALA4338968 | A | Half life in Sprague-Dawley rat at 1 mg/kg, iv or 2 mg/kg, po | Rattus norvegicus | 4 | organism-based format | Scientific Literature |
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