| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4333246 | B | Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assay | Homo sapiens | 36 | assay format | Scientific Literature | ||
| 2. | ALA4333251 | B | Binding affinity to human wild-type AAK1 (G25 to L333 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 3. | ALA4333252 | B | Binding affinity to human phosphorylated ABL1 E255K mutant (S229 to K512 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 4. | ALA4333253 | B | Binding affinity to human non-phosphorylated ABL1 F317I mutant (S229 to K512 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 5. | ALA4333254 | B | Binding affinity to human phosphorylated ABL1 F317I mutant (S229 to K512 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 6. | ALA4333255 | B | Binding affinity to human non-phosphorylated ABL1 F317L mutant (S229 to K512 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 7. | ALA4333256 | B | Binding affinity to human phosphorylated ABL1 F317L mutant (S229 to K512 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 8. | ALA4333257 | B | Binding affinity to human non-phosphorylated ABL1 H396P mutant (S229 to K512 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 9. | ALA4333258 | B | Binding affinity to human phosphorylated ABL1 H396P mutant (S229 to K512 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 10. | ALA4333259 | B | Binding affinity to human phosphorylated ABL1 M351T mutant (S229 to K512 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 11. | ALA4333260 | B | Binding affinity to human non-phosphorylated ABL1 Q252H mutant (S229 to K512 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 12. | ALA4333261 | B | Binding affinity to human phosphorylated ABL1 Q252H mutant expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 13. | ALA4333262 | B | Binding affinity to human non-phosphorylated ABL1 T315I mutant (S229 to K512 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA4333263 | B | Binding affinity to human phosphorylated ABL1 T315I mutant (S229 to K512 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA4333264 | B | Binding affinity to human phosphorylated ABL1 Y253F mutant (S229 to K512 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 16. | ALA4333265 | B | Binding affinity to wild-type human non-phosphorylated ABL1 (S229 to K512 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA4333266 | B | Binding affinity to wild-type human phosphorylated ABL1 (S229 to K512 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 18. | ALA4333267 | B | Binding affinity to wild-type human ABL2 (A248 to G542 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 19. | ALA4333268 | B | Binding affinity to wild-type human ACVR1 (C188 to C509 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 20. | ALA4333269 | B | Binding affinity to wild-type human ACVR1B (S187 to I505 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | assay format | Scientific Literature |
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