| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4330014 | B | Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris strain X-33 using Ac-YRSR-pNA as substrate preincubated for 30 mins followed by substrate addition and measured for 7 mins by spectrophotometric method | Homo sapiens | 3 | assay format | Scientific Literature | ||
| 2. | ALA4330015 | A | Stability in human serum at 200 uM up to 24 hrs by RP-HPLC analysis | Homo sapiens | 3 | cell-free format | Scientific Literature | ||
| 3. | ALA4330016 | B | Inhibition of KLK4 (unknown origin) expressed in sf9 cells using Ac-FVQR-pNA as substrate preincubated for 30 mins followed by substrate addition and measured for 7 mins by spectrophotometric method | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 4. | ALA4330017 | B | Inhibition of plasmin (unknown origin) using Ac-RM(O2)YR-pNA as substrate preincubated for 30 mins followed by substrate addition and measured for 7 mins by spectrophotometric method | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 5. | ALA4330019 | B | Inhibition of KLK7 (unknown origin) expressed in Pichia pastoris strain X-33 using KHLY-pNA as substrate preincubated for 30 mins followed by substrate addition and measured for 7 mins by spectrophotometric method | Homo sapiens | 3 | assay format | Scientific Literature | ||
| 6. | ALA4330020 | B | Inhibition of KLK14 (unknown origin) expressed in sf9 cells using Ac-YANR-pNA as substrate preincubated for 30 mins followed by substrate addition and measured for 7 mins by spectrophotometric method | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 7. | ALA4330021 | B | Inhibition of factor 10a (unknown origin) using Ac-QRSR-pNA as substrate preincubated for 30 mins followed by substrate addition and measured for 7 mins by spectrophotometric method | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 8. | ALA4330022 | B | Inhibition of thrombin (unknown origin) using Bz-FVR-pNA as substrate preincubated for 30 mins followed by substrate addition and measured for 7 mins by spectrophotometric method | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 9. | ALA4330023 | B | Inhibition of plasma kallikrein (unknown origin) using Ac-NLTR-pNA as substrate preincubated for 30 mins followed by substrate addition and measured for 7 mins by spectrophotometric method | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 10. | ALA4330024 | B | Inhibition of trypsin (unknown origin) using Bz-FVR-pNA as substrate preincubated for 30 mins followed by substrate addition and measured for 7 mins by spectrophotometric method | Homo sapiens | 2 | protein format | Scientific Literature | ||
| 11. | ALA4330025 | B | Inhibition of factor 12a (unknown origin) using Ac-QRFR-pNA as substrate preincubated for 30 mins followed by substrate addition and measured for 7 mins by spectrophotometric method | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 12. | ALA4330026 | B | Selectivity ratio of Ki for KLK5 (unknown origin) expressed in Pichia pastoris strain X-33 to Ki for KLK4 (unknown origin) expressed in sf9 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 13. | ALA4330027 | B | Selectivity ratio of Ki for KLK7 (unknown origin) expressed in Pichia pastoris strain X-33 to Ki for KLK4 (unknown origin) expressed in sf9 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 14. | ALA4330028 | B | Selectivity ratio of Ki for KLK14 (unknown origin) expressed in sf9 cells to Ki for KLK4 (unknown origin) expressed in sf9 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 15. | ALA4330029 | B | Selectivity ratio of Ki for plasmin (unknown origin) to Ki for KLK4 (unknown origin) expressed in sf9 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 16. | ALA4330030 | B | Selectivity ratio of Ki for factor 12a (unknown origin) to Ki for KLK4 (unknown origin) expressed in sf9 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA4330031 | B | Selectivity ratio of Ki for thrombin (unknown origin) to Ki for KLK4 (unknown origin) expressed in sf9 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 18. | ALA4330032 | B | Selectivity ratio of Ki for plasma kallikrein (unknown origin) to Ki for KLK4 (unknown origin) expressed in sf9 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 19. | ALA4330033 | B | Selectivity ratio of Ki for factor 10a (unknown origin) to Ki for KLK4 (unknown origin) expressed in sf9 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 20. | ALA4330034 | A | Drug uptake in human HeLa cells at 4 uM using Alexa Fluor 488 conjugated test compound after 1 hr by trypan blue dye based flow cytometry relative to HIV-Tat | Homo sapiens | 5 | cell-based format | Scientific Literature |
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