| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4427614 | B | Inhibition of ALK5 (unknown origin) using fluorescein-labeled peptide substrate incubated for 90 mins by TR-FRET assay | Homo sapiens | 19 | ALA4425174 | single protein format | Scientific Literature | |
| 2. | ALA4427615 | B | Inhibition of ALK5 in TGF beta1-stimulated HEK293T cells by SMAD binding element-driven beta lactamase reporter gene assay | Homo sapiens | 15 | ALA4425174 | assay format | Scientific Literature | |
| 3. | ALA4427616 | A | Inhibition of CYP1A2 (unknown origin) | Homo sapiens | 18 | ALA4425174 | single protein format | Scientific Literature | |
| 4. | ALA4427618 | A | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 18 | ALA4425174 | single protein format | Scientific Literature | |
| 5. | ALA4427619 | A | Intrinsic clearance in rat liver microsomes | Rattus norvegicus | 18 | ALA4425174 | microsome format | Scientific Literature | |
| 6. | ALA4427620 | A | Oral bioavailability in rat | Rattus norvegicus | 4 | ALA4425174 | organism-based format | Scientific Literature | |
| 7. | ALA4427621 | B | Inhibition of human ERG at 10 uM relative to control | Homo sapiens | 1 | ALA4425174 | single protein format | Scientific Literature | |
| 8. | ALA4427622 | B | Inhibition of ABL1 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4425174 | single protein format | Scientific Literature | |
| 9. | ALA4427623 | B | Inhibition of AKT1 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4425174 | single protein format | Scientific Literature | |
| 10. | ALA4427624 | B | Inhibition of Aurora A (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4425174 | single protein format | Scientific Literature | |
| 11. | ALA4427625 | B | Inhibition of BRAF (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4425174 | single protein format | Scientific Literature | |
| 12. | ALA4427626 | B | Inhibition of CDK1/Cyclin B (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4425174 | protein complex format | Scientific Literature | |
| 13. | ALA4427627 | B | Inhibition of CDK2/Cyclin A (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4425174 | protein complex format | Scientific Literature | |
| 14. | ALA4427628 | B | Inhibition of CDK5/p25 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4425174 | protein complex format | Scientific Literature | |
| 15. | ALA4427629 | B | Inhibition of CHK1 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4425174 | single protein format | Scientific Literature | |
| 16. | ALA4427630 | B | Inhibition of CHK2 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4425174 | single protein format | Scientific Literature | |
| 17. | ALA4427631 | B | Inhibition of CLK1 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4425174 | single protein format | Scientific Literature | |
| 18. | ALA4427632 | B | Inhibition of CLK2 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4425174 | single protein format | Scientific Literature | |
| 19. | ALA4427633 | B | Inhibition of CSK (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4425174 | single protein format | Scientific Literature | |
| 20. | ALA4427634 | B | Inhibition of EGFR (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4425174 | single protein format | Scientific Literature |
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