# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4424973 | B | Inhibition of recombinant human DAGLalpha expressed in COS7 cells using [14C]-oleoyl-2-arachidonoyl-glycerol as substrate measured after 20 mins by beta-counting method | Homo sapiens | 11 | ALA4422692 | cell-based format | Scientific Literature | |
2. | ALA4424974 | B | Inhibition of recombinant human DAGLalpha expressed in COS7 cells at 50 uM using [14C]-oleoyl-2-arachidonoyl-glycerol as substrate measured after 20 mins by beta-counting method relative to control | Homo sapiens | 8 | ALA4422692 | cell-based format | Scientific Literature | |
3. | ALA4424976 | B | Inhibition of MAGL in African green monkey COS cell homogenates using [3H]-arachidonoylglycerol as substrate measured after 20 mins by scintillation counting method | Chlorocebus aethiops | 10 | ALA4422692 | tissue-based format | Scientific Literature | |
4. | ALA4424978 | B | Inhibition of MAGL in African green monkey COS cell homogenates at 50 uM using [3H]-arachidonoylglycerol as substrate measured after 20 mins by scintillation counting method relative to control | Chlorocebus aethiops | 5 | ALA4422692 | tissue-based format | Scientific Literature | |
5. | ALA4424979 | B | Inhibition of FAAH in rat brain membranes using [14C]-AEA as substrate measured after 30 mins by scintillation counting method | Rattus norvegicus | 10 | ALA4422692 | cell membrane format | Scientific Literature | |
6. | ALA4424981 | B | Inhibition of FAAH in rat brain membranes at 100 uM using [14C]-AEA as substrate measured after 30 mins by scintillation counting method relative to control | Rattus norvegicus | 5 | ALA4422692 | cell membrane format | Scientific Literature | |
7. | ALA4424982 | B | Inhibition of recombinant human NAAA expressed in HEK293 cells using [14C]-N-palmitoylethanolamine as substrate measured after 30 mins by beta-counting method | Homo sapiens | 10 | ALA4422692 | cell-based format | Scientific Literature | |
8. | ALA4424984 | B | Inhibition of recombinant human NAAA expressed in HEK293 cells at 50 uM using [14C]-N-palmitoylethanolamine as substrate measured after 30 mins by beta-counting method relative to control | Homo sapiens | 6 | ALA4422692 | cell-based format | Scientific Literature | |
9. | ALA4424985 | F | Inhibition of [14C]-AEA uptake in rat RBL2H3 cells by scintillation counting method | Rattus norvegicus | 10 | ALA4422692 | cell-based format | Scientific Literature | |
10. | ALA4424986 | F | Inhibition of [14C]-AEA uptake in rat RBL2H3 cells at 25 uM by scintillation counting method relative to control | Rattus norvegicus | 10 | ALA4422692 | cell-based format | Scientific Literature | |
11. | ALA4842433 | B | Inhibition of human LDHB assessed as reduction in lactate production using pyruvate as substrate at 10 uM in presence of NADH by spectrophotometric analysis relative to control | Homo sapiens | 18 | ALA4842310 | single protein format | Scientific Literature |