# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4371895 | Binding | Inhibition of mouse GAT1 expressed in HEK cells assessed as reduction in [3H]GABA uptake by measuring remaining [3H]GABA uptake levels preincubated for 25 mins followed by [3H]GABA addition and measured after 4 mins by microbeta liquid scintillation counting analysis | Mus musculus | 3 | ALA4371022 | cell-based format | Scientific Literature | |
2. | ALA4371898 | Binding | Inhibition of mouse GAT2 expressed in HEK cells assessed as reduction in [3H]GABA uptake at 100 uM by measuring remaining [3H]GABA uptake levels preincubated for 25 mins followed by [3H]GABA addition and measured after 4 mins by microbeta liquid scintillation counting analysis | Mus musculus | 3 | ALA4371022 | cell-based format | Scientific Literature | |
3. | ALA4371900 | Binding | Inhibition of mouse GAT3 expressed in HEK cells assessed as reduction in [3H]GABA uptake at 100 uM by measuring remaining [3H]GABA uptake levels preincubated for 25 mins followed by [3H]GABA addition and measured after 4 mins by microbeta liquid scintillation counting analysis | Mus musculus | 1 | ALA4371022 | cell-based format | Scientific Literature | |
4. | ALA4371901 | Binding | Inhibition of mouse GAT4 expressed in HEK cells assessed as reduction in [3H]GABA uptake by measuring remaining [3H]GABA uptake levels preincubated for 25 mins followed by [3H]GABA addition and measured after 4 mins by microbeta liquid scintillation counting analysis | Mus musculus | 4 | ALA4371022 | cell-based format | Scientific Literature | |
5. | ALA4371902 | Binding | Inhibition of human GAT3 expressed in COS7 cells assessed as reduction in [2H6]GABA uptake preincubated for 25 mins followed by [2H6]GABA addition and measured after 6 mins by LC-MS/MS analysis | Homo sapiens | 4 | ALA4371022 | cell-based format | Scientific Literature | |
6. | ALA4767574 | Binding | Inhibition of mouse GTA 1 receptor | Mus musculus | 8 | ALA4765247 | single protein format | Scientific Literature | |
7. | ALA4767575 | Binding | Inhibition of mouse GTA 2 receptor | Mus musculus | 8 | ALA4765247 | single protein format | Scientific Literature | |
8. | ALA4767576 | Binding | Inhibition of mouse GTA 3 receptor | Mus musculus | 8 | ALA4765247 | single protein format | Scientific Literature | |
9. | ALA4767577 | Binding | Inhibition of mouse GTA4 receptor | Mus musculus | 8 | ALA4765247 | single protein format | Scientific Literature |