| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4338950 | B | Inhibition of recombinant N-terminal FLAG/His-tagged SMYD3 (unknown origin) expressed in baculovirus infected insect cells using 3H-SAM as substrate assessed as 3H-MEKK2 methylation incubated for 40 mins by scintillation proximity assay | Homo sapiens | 49 | cell-based format | Scientific Literature | ||
| 2. | ALA4338951 | B | Inhibition of recombinant SMYD3 (unknown origin) transfected in human HEK293 cells assessed as reduction in MEKK2 methylation incubated for 24 hrs by cellular mechanistic assay | Homo sapiens | 49 | cell-based format | Scientific Literature | ||
| 3. | ALA4338952 | P | Solubility of compound by CLND method | 47 | small-molecule physicochemical format | Scientific Literature | |||
| 4. | ALA4338953 | A | Permeability of compound | 44 | assay format | Scientific Literature | |||
| 5. | ALA4338957 | B | Inhibition of recombinant SMYD3 in human A549 cells assessed as reduction in ERK1/2 phosphorylation at 30 uM preincubated for 72 hrs followed by incubated in serum free for 24 hrs by Western blot analysis | Homo sapiens | 3 | cell-based format | Scientific Literature |
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