| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4431786 | Binding | Inhibition of recombinant Toxoplasma gondii CDPK1 using Biotin-C6-PLARTLSVAGLPGKK as substrate after 90 mins in presence of ATP by luciferase reporter gene assay | Toxoplasma gondii | 34 | ALA4431312 | single protein format | Scientific Literature | |
| 2. | ALA4431787 | Binding | Inhibition of chicken Src using AcEIYGEFKKK as substrate after 90 mins in presence of ATP by luciferase reporter gene assay | Gallus gallus | 32 | ALA4431312 | single protein format | Scientific Literature | |
| 3. | ALA4431789 | ADME | Growth inhibition of human HepG2 cells after 48 hrs by Alamar blue assay | Homo sapiens | 30 | ALA4431312 | cell-based format | Scientific Literature | |
| 4. | ALA4431790 | ADME | Growth inhibition of human CRL8155 cells after 48 hrs by Alamar blue assay | Homo sapiens | 31 | ALA4431312 | assay format | Scientific Literature | |
| 5. | ALA4431791 | Binding | Inhibition of human ERG | Homo sapiens | 27 | ALA4431312 | single protein format | Scientific Literature | |
| 6. | ALA4431792 | Functional | Antiparasitic activity against Toxoplasma gondii infected in human foreskin fibroblasts assessed as reduction of parasite invasion after 44 hrs by beta-galactosidase reporter gene assay | Toxoplasma gondii | 30 | ALA4431312 | organism-based format | Scientific Literature | |
| 7. | ALA4431794 | Physicochemical | Solubility of the compound in phosphate buffered saline at pH 6.5 by HPLC/UV analysis | 9 | ALA4431312 | small-molecule physicochemical format | Scientific Literature | ||
| 8. | ALA4431795 | ADME | Tmax in BALB/c mouse plasma at 10 mg/kg administered via oral gavage by LC/MS analysis | Mus musculus | 9 | ALA4431312 | organism-based format | Scientific Literature | |
| 9. | ALA4431796 | ADME | Cmax in BALB/c mouse plasma at 10 mg/kg administered via oral gavage by LC/MS analysis | Mus musculus | 9 | ALA4431312 | organism-based format | Scientific Literature | |
| 10. | ALA4431797 | ADME | AUC (0 to infinity) in BALB/c mouse plasma at 10 mg/kg administered via oral gavage by LC/MS analysis | Mus musculus | 9 | ALA4431312 | organism-based format | Scientific Literature | |
| 11. | ALA4431798 | ADME | Half life in BALB/c mouse plasma at 10 mg/kg administered via oral gavage by LC/MS analysis | Mus musculus | 9 | ALA4431312 | organism-based format | Scientific Literature | |
| 12. | ALA4431799 | ADME | Clearance in BALB/c mouse plasma at 10 mg/kg administered via oral gavage by LC/MS analysis | Mus musculus | 9 | ALA4431312 | organism-based format | Scientific Literature | |
| 13. | ALA4774309 | Binding | Inhibition of recombinant FLAG-tagged PKD1 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo assay | Homo sapiens | 9 | ALA4765437 | cell-based format | Scientific Literature | |
| 14. | ALA4774310 | Binding | Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo assay | Homo sapiens | 9 | ALA4765437 | cell-based format | Scientific Literature | |
| 15. | ALA4774311 | Binding | Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo assay | Homo sapiens | 9 | ALA4765437 | cell-based format | Scientific Literature | |
| 16. | ALA4774321 | Functional | Antiproliferative activity against human LN-229 cells assessed as reduction in cell viability incubated for 72 hrs by IncuCyte live-cell automated imaging analysis | Homo sapiens | 7 | ALA4765437 | cell-based format | Scientific Literature | |
| 17. | ALA4774322 | Functional | Antiproliferative activity against human CAPAN-1 cells assessed as reduction in cell viability incubated for 72 hrs by IncuCyte live-cell automated imaging analysis | Homo sapiens | 7 | ALA4765437 | cell-based format | Scientific Literature | |
| 18. | ALA4774323 | Functional | Antiproliferative activity against human HCT-116 cells assessed as reduction in cell viability incubated for 72 hrs by IncuCyte live-cell automated imaging analysis | Homo sapiens | 7 | ALA4765437 | cell-based format | Scientific Literature | |
| 19. | ALA4774324 | Functional | Antiproliferative activity against human NCI-H460 cells assessed as reduction in cell viability incubated for 72 hrs by IncuCyte live-cell automated imaging analysis | Homo sapiens | 7 | ALA4765437 | cell-based format | Scientific Literature | |
| 20. | ALA4774325 | Functional | Antiproliferative activity against human DND41 cells assessed as reduction in cell viability incubated for 72 hrs by IncuCyte live-cell automated imaging analysis | Homo sapiens | 7 | ALA4765437 | cell-based format | Scientific Literature |
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