# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4312045 | B | Inhibition of BRD2 (unknown origin) by TR-FRET assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
2. | ALA4312046 | B | Inhibition of BRD3 (unknown origin) by TR-FRET assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
3. | ALA4312047 | B | Inhibition of BRD4 (unknown origin) by TR-FRET assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
4. | ALA4312048 | B | Inhibition of BRD4 in human MX1 cells assessed as decrease in cell proliferation after 3 days by Celltiter-Glo assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
5. | ALA4312049 | B | Inhibition of BRD4 in human H1229 cells transfected with HPV-E2 assessed as transrepression of HPV-long control region by luciferase reporter assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
6. | ALA4312050 | A | Permeability of compound in 5% DMSO after 7 hrs by PAMPA | 40 | assay format | Scientific Literature | |||
7. | ALA4312051 | A | Ratio of drug concentration in unbound HEK293 cell to media | 13 | assay format | Scientific Literature | |||
8. | ALA4312074 | B | Inhibition of BRD4 in human MX1 cells assessed as decrease in cell proliferation after 3 days by Celltiter-Glo assay relative to parent compound | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
9. | ALA4312075 | B | Inhibition of BRD4 in luciferase expressing human H1229 cells transfected with HPV-E2 assessed as transrepression of HPV-long control region by luciferase reporter assay relative to parent compound | Homo sapiens | 5 | assay format | Scientific Literature |