| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4372793 | B | Displacement of [3H]U-69,593 from KOR in guinea pig brain membranes after 120 mins by scintillation counting method | Cavia porcellus | 15 | cell membrane format | Scientific Literature | ||
| 2. | ALA4372794 | A | Displacement of [3H]DAMGO from MOR in guinea pig brain membranes after 120 mins by scintillation counting method | Cavia porcellus | 8 | cell membrane format | Scientific Literature | ||
| 3. | ALA4372795 | B | Displacement of [3H]DPDPE from DOR in Sprague-Dawley rat brain membranes after 120 mins by scintillation counting method | Rattus norvegicus | 13 | cell membrane format | Scientific Literature | ||
| 4. | ALA4372796 | B | Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membranes after 120 mins by scintillation counting method | Cavia porcellus | 5 | cell membrane format | Scientific Literature | ||
| 5. | ALA4372797 | B | Displacement of [3H]DTG from sigma2 receptor in rat liver membranes after 120 mins by scintillation counting method | Rattus norvegicus | 3 | cell membrane format | Scientific Literature | ||
| 6. | ALA4372798 | A | Displacement of [3H]DAMGO from MOR in guinea pig brain membranes at 1 uM after 120 mins by scintillation counting method relative to control | Cavia porcellus | 13 | cell membrane format | Scientific Literature | ||
| 7. | ALA4372799 | B | Displacement of [3H]DPDPE from DOR in Sprague-Dawley rat brain membranes at 1 uM after 120 mins by scintillation counting method relative to control | Rattus norvegicus | 13 | cell membrane format | Scientific Literature | ||
| 8. | ALA4372800 | B | Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membranes at 1 uM after 120 mins by scintillation counting method relative to control | Cavia porcellus | 13 | cell membrane format | Scientific Literature | ||
| 9. | ALA4372801 | B | Displacement of [3H]DTG from sigma2 receptor in rat liver membranes at 1 uM after 120 mins by scintillation counting method relative to control | Rattus norvegicus | 13 | cell membrane format | Scientific Literature | ||
| 10. | ALA4372802 | B | Displacement of [3H]diprenorphine from human KOR expressed in HEK293T cell membranes after 120 mins by scintillation counting method | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 11. | ALA4372803 | F | Agonist activity at human KOR expressed in HEK293T cells assessed as inhibition of Galphai-mediated cAMP accumulation after 15 mins by microbeta counting assay relative to salvinorin A | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 12. | ALA4372804 | F | Agonist activity at human KOR expressed in HEK293T cells assessed as inhibition of Galphai-mediated cAMP accumulation after 15 mins by microbeta counting assay | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 13. | ALA4372809 | B | Ratio of Ki for displacement of [3H]diprenorphine from human KOR expressed in HEK293T cell membranes to Ki for displacement of [3H]U-69,593 from KOR in guinea pig brain membranes | 8 | cell-based format | Scientific Literature | |||
| 14. | ALA4372810 | B | Agonist activity at Tango-KOR (unknown origin) expressed in HTLA cells harboring TEV-fused-beta-arrestin 2 assessed as increase in beta arrestin 2 recruitment after overnight incubation by BrightGlo reagent based assay | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 15. | ALA4372811 | B | Agonist activity at Tango-KOR (unknown origin) expressed in HTLA cells harboring TEV-fused-beta-arrestin 2 assessed as increase in beta arrestin 2 recruitment after overnight incubation by BrightGlo reagent based assay relative to salvinorin A | Homo sapiens | 9 | cell-based format | Scientific Literature |
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