# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4427931 | Binding | Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assay | Homo sapiens | 20 | ALA4425189 | single protein format | Scientific Literature | |
2. | ALA4427945 | Binding | Inhibition of KDM5A in human PC9 cells assessed as increase in H3K4me3 levels preincubated for 4 days measured up to 24 hrs by ELISA | Homo sapiens | 2 | ALA4425189 | cell-based format | Scientific Literature | |
3. | ALA4427947 | Binding | Inhibition of of KDM5 in human U2OS cells assessed as effect on in H3K4me3 levels at 15 uM by Western blot analysis | Homo sapiens | 1 | ALA4425189 | cell-based format | Scientific Literature | |
4. | ALA4427951 | Functional | Induction of KDM5A transcription levels in human U2OS cells at 15 uM by Western blot analysis | Homo sapiens | 1 | ALA4425189 | cell-based format | Scientific Literature | |
5. | ALA4427952 | Functional | Induction of KDM5B transcription levels in human U2OS cells at 15 uM by Western blot analysis | Homo sapiens | 1 | ALA4425189 | cell-based format | Scientific Literature | |
6. | ALA4427953 | Functional | Induction of KDM5C transcription levels in human U2OS cells at 15 uM by Western blot analysis | Homo sapiens | 1 | ALA4425189 | cell-based format | Scientific Literature |