| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4334911 | B | Inhibition of human GSK-3alpha S449A mutant (2 to end residues) at 10 uM using phospho GS2 peptide as substrate after 40 mins in presence of [gamma-33ATP] by scintillation counting method relative to control | Homo sapiens | 80 | single protein format | Scientific Literature | ||
| 2. | ALA4334912 | B | Inhibition of human GSK-3alpha S449A mutant (2 to end residues) using phospho GS2 peptide as substrate after 40 mins in presence of [gamma-33ATP] by scintillation counting method | Homo sapiens | 54 | single protein format | Scientific Literature | ||
| 3. | ALA4334913 | A | Inhibition of human GSK-3beta H350L mutant (2 to end residues) at 10 uM using phospho GS2 peptide as substrate after 40 mins by [gamma-33ATP] radiometric assay relative to control | Homo sapiens | 48 | single protein format | Scientific Literature | ||
| 4. | ALA4334914 | A | Inhibition of human GSK-3beta H350L mutant (2 to end residues) at 10 uM using phospho GS2 peptide as substrate after 40 mins by [gamma-33ATP] radiometric assay | Homo sapiens | 48 | single protein format | Scientific Literature | ||
| 5. | ALA4334915 | B | Selectivity index, ratio of IC50 for inhibition of human GSK-3beta H350L mutant (2 to end residues) to IC50 for inhibition of human GSK-3alpha S449A mutant (2 to end residues) | Homo sapiens | 3 | assay format | Scientific Literature |
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