# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4397555 | Binding | Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assay | Mus musculus | 23 | ALA4396875 | cell-based format | Scientific Literature | |
2. | ALA4397556 | Binding | Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assay | Homo sapiens | 23 | ALA4396875 | cell-based format | Scientific Literature | |
3. | ALA4397557 | Binding | Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as activation of GalphaS incubated for 5 mins in presence of coelenterazine 400a by BRET assay relative to isoprenaline | Homo sapiens | 10 | ALA4396875 | cell-based format | Scientific Literature | |
4. | ALA4397558 | Binding | Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as activation of GalphaS incubated for 5 mins in presence of coelenterazine 400a by BRET assay | Homo sapiens | 7 | ALA4396875 | cell-based format | Scientific Literature | |
5. | ALA4397559 | Binding | Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment incubated for 5 mins in presence of coelenterazine 400a by BRET assay relative to isoprenaline | Homo sapiens | 10 | ALA4396875 | cell-based format | Scientific Literature | |
6. | ALA4397560 | Binding | Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment incubated for 5 mins in presence of coelenterazine 400a by BRET assay | Homo sapiens | 6 | ALA4396875 | cell-based format | Scientific Literature | |
7. | ALA4397561 | Binding | Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment incubated for 5 mins in presence of GRK2 and coelenterazine 400a by BRET assay relative to isoprenaline | Homo sapiens | 10 | ALA4396875 | cell-based format | Scientific Literature | |
8. | ALA4397562 | Binding | Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment incubated for 5 mins in presence of GRK2 and coelenterazine 400a by BRET assay | Homo sapiens | 6 | ALA4396875 | cell-based format | Scientific Literature | |
9. | ALA4397563 | Binding | Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment incubated for 5 mins in presence of GRK5 and coelenterazine 400a by BRET assay relative to isoprenaline | Homo sapiens | 10 | ALA4396875 | cell-based format | Scientific Literature | |
10. | ALA4397564 | Binding | Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment incubated for 5 mins in presence of GRK5 and coelenterazine 400a by BRET assay | Homo sapiens | 7 | ALA4396875 | cell-based format | Scientific Literature | |
11. | ALA4397565 | Binding | Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as activation of GalphaS incubated for 5 mins in presence of coelenterazine 400a by BRET assay relative to isoprenaline | Homo sapiens | 10 | ALA4396875 | cell-based format | Scientific Literature | |
12. | ALA4397566 | Binding | Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as activation of GalphaS incubated for 5 mins in presence of coelenterazine 400a by BRET assay | Homo sapiens | 7 | ALA4396875 | cell-based format | Scientific Literature | |
13. | ALA4397567 | Binding | Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment incubated for 5 mins in presence of coelenterazine 400a by BRET assay relative to isoprenaline | Homo sapiens | 10 | ALA4396875 | cell-based format | Scientific Literature | |
14. | ALA4397569 | Binding | Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment incubated for 5 mins in presence of GSK2 and coelenterazine 400a by BRET assay relative to isoprenaline | Homo sapiens | 10 | ALA4396875 | cell-based format | Scientific Literature | |
15. | ALA4397571 | Binding | Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment incubated for 5 mins in presence of GSK5 and coelenterazine 400a by BRET assay relative to isoprenaline | Homo sapiens | 10 | ALA4396875 | cell-based format | Scientific Literature | |
16. | ALA4397572 | Binding | Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment incubated for 5 mins in presence of GSK5 and coelenterazine 400a by BRET assay | Homo sapiens | 7 | ALA4396875 | cell-based format | Scientific Literature |