| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4612974 | B | Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintillation counting method | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 2. | ALA4612975 | F | Antagonist activity at human CGRP receptor in human SK-N-MC cells assessed as inhibition of CGRP-induced cAMP production preincubated for 30 mins followed by CGRP addition and measured after 30 mins by HTRF assay | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 3. | ALA4612976 | P | Thermodynamic solubility of the compound at pH 6 | 9 | small-molecule physicochemical format | Scientific Literature | |||
| 4. | ALA4612977 | P | Thermodynamic solubility of the compound at pH 7.4 | 9 | small-molecule physicochemical format | Scientific Literature | |||
| 5. | ALA4612979 | A | Clearance in rat at 0.5 mg/kg, iv | Rattus norvegicus | 1 | organism-based format | Scientific Literature |
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