| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4612600 | B | Inhibition of recombinant human Lp-PLA2 (47 to 429 residues) expressed in Escherichia coli RosettaTM2 (DE3) pLysS | Homo sapiens | 10 | ALA4610113 | assay format | Scientific Literature | |
| 2. | ALA4612601 | B | Selectivity index, ratio of IC50 for full-length PLA2VIIB (unknown origin) to IC50 for human Lp-PLA2 (47 to 429 residues) expressed in Escherichia coli RosettaTM2 (DE3) pLysS | Homo sapiens | 4 | ALA4610113 | assay format | Scientific Literature | |
| 3. | ALA4612608 | B | Time dependent inhibition of recombinant human Lp-PLA2 (47 to 429 residues) expressed in Escherichia coli RosettaTM2 (DE3) pLysS assessed as Kinact/Ki ratio | Homo sapiens | 2 | ALA4610113 | assay format | Scientific Literature | |
| 4. | ALA4612609 | B | Inhibition of full-length PLA2VIIB (unknown origin) expressed in Escherichia coli RosettaTM2 (DE3) pLysS at 50 uM relative to control | Homo sapiens | 1 | ALA4610113 | assay format | Scientific Literature | |
| 5. | ALA4612610 | B | Binding affinity to Lp-PLA2 in HEK293T cell lysates up to 50 uM by FP-TAMRA probe based activity-based protein profiling assay | Homo sapiens | 1 | ALA4610113 | cell-based format | Scientific Literature | |
| 6. | ALA4612611 | B | Binding affinity to recombinant human Lp-PLA2 (47 to 429 residues) in HEK293T cell lysates up to 50 uM by FP-TAMRA probe based activity-based protein profiling assay | Homo sapiens | 1 | ALA4610113 | cell-based format | Scientific Literature | |
| 7. | ALA4612615 | B | Inhibition of recombinant human Lp-PLA2 (47 to 429 residues) in HEK293T cell lysates at 2 uM in presence of 8-BODIPY by gel-based competitive ABPP analysis | Homo sapiens | 1 | ALA4610113 | cell-based format | Scientific Literature | |
| 8. | ALA4612616 | B | Inhibition of recombinant human Lp-PLA2 (47 to 429 residues) in HEK293T cell lysates at 2 uM in presence of 8-RH by gel-based competitive ABPP analysis | Homo sapiens | 1 | ALA4610113 | cell-based format | Scientific Literature | |
| 9. | ALA5127352 | B | Inhibition of recombinant human Lp-PLA2 using 2-thio-PAF as substrate preincubated for 30 mins followed by substrate addition | Homo sapiens | 2 | ALA5126516 | single protein format | Scientific Literature |
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